SCHEMBL6109657

SCHEMBL6109657

COc1ccc(-c2cccs2)c(OC)c1C(=O)C=Cc1cccc(OC(C)(C)C(=O)O)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 15/20 0.50
ABCG2 Q9UNQ0 1/20 0.44
MEN1 O00255 2/20 0.43
ALDH1A1 P00352 2/20 0.43
TP53 P04637 2/20 0.43
CYP3A4 P08684 2/20 0.43
MAPT P10636 2/20 0.43
HPGD P15428 2/20 0.43
KMT2A Q03164 2/20 0.43
HSD17B10 Q99714 2/20 0.43
KDM4E B2RXH2 1/20 0.43
CASP7 P55210 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MAPK1 P28482 1/20 0.43
ABCB1 P08183 1/20 0.41
BCHE P06276 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6109489 0.90 TNFRSF1A (0.50) TNFRSF1AMEN1ALDH1A1TP53CYP3A4
SCHEMBL6110383 0.83 TNFRSF1A (0.58) TNFRSF1AABCG2MEN1ALDH1A1TP53
SCHEMBL25208831 0.83 TNFRSF1A (0.58) TNFRSF1AABCG2MEN1ALDH1A1TP53
SCHEMBL6093024 0.80 PPARG (0.42) TNFRSF1AMAPTKDM4E
SCHEMBL6091213 0.79 TNFRSF1A (0.42) TNFRSF1AMEN1ALDH1A1MAPTHPGD
SCHEMBL6109512 0.78 TNFRSF1A (0.58) TNFRSF1AABCG2MEN1ALDH1A1TP53
SCHEMBL6111525 0.75 TNFRSF1A (0.81) TNFRSF1A
SCHEMBL6093002 0.75 PPARA (0.42) TNFRSF1AMAPTKDM4EMAPK1
SCHEMBL6091494 0.74 TNFRSF1A (0.44) TNFRSF1AMEN1ALDH1A1CYP3A4MAPT
SCHEMBL6111017 0.70 TNFRSF1A (0.49) TNFRSF1AMEN1ALDH1A1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006004903-A2 1,2-BIS-(SUBSTITUTED-PHENYL)-2-PROPEN-1-ONES AND PHARMACEUTICAL COMPOSITIONS THEREOF ATHEROGENICS, INC. (US) 2006-01-12 WO claimed
WO-2006004903-A2 1,2-BIS-(SUBSTITUTED-PHENYL)-2-PROPEN-1-ONES AND PHARMACEUTICAL COMPOSITIONS THEREOF ATHEROGENICS, INC. (US) 2006-01-12 WO disclosed