SCHEMBL6110464

SCHEMBL6110464

Cc1ccc2c(N3CC[C@H](COC(N)=O)C3)nc(-c3ccccc3O)nc2c1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.49
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
SMAD3 P84022 1/20 0.43
MAPT P10636 4/20 0.41
ALDH1A1 P00352 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
TSHR P16473 2/20 0.41
HIF1A Q16665 1/20 0.41
KDM4E B2RXH2 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
CHRM3 P20309 4/20 0.38
TP53 P04637 1/20 0.38
ADORA2A P29274 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6110469 1.00 CHEK2 (0.49) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL1084868 0.89 CHEK2 (0.54) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL1621898 0.86 CHEK2 (0.55) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL1624407 0.86 CHEK2 (0.55) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL1621902 0.86 CHEK2 (0.55) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL1084747 0.85 SMAD3 (0.51) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL5499288 0.84 CHEK2 (0.50) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL5499286 0.84 CHEK2 (0.50) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL4011379 0.84 CHEK2 (0.55) CHEK2KMT2AMEN1SMAD3MAPT
SCHEMBL4014734 0.84 CHEK2 (0.55) CHEK2KMT2AMEN1SMAD3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006028904-A9 QUINAZOLINES USEFUL AS MODULATORS OF ION CHANNELS VERTEX PHARMA (US) 2006-06-22 WO disclosed