SCHEMBL6120195

SCHEMBL6120195

C=CCN(C)CCN(c1cc2oc(-c3ccc(F)cc3)c(C(=O)NC)c2cc1OC(C)C)S(C)(=O)=O

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 3/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2C19 P33261 2/20 0.46
KCNH2 Q12809 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2837508 0.93 CYP2C9 (0.50) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6120324 0.88 CYP3A4 (0.49) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2838885 0.88 CYP3A4 (0.51) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2837509 0.87 CYP3A4 (0.50) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2839906 0.86 CYP3A4 (0.52) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL6119339 0.86 CYP3A4 (0.49) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2843854 0.84 CYP3A4 (0.51) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2835951 0.84 CYP3A4 (0.51) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL2841638 0.84 CYP3A4 (0.51) CYP2C9CYP3A4CYP2C19KCNH2
SCHEMBL3397081 0.84 CYP3A4 (0.48) CYP2C9CYP3A4CYP2C19KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012067663-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-05-24 WO disclosed