Epristeride

Epristeride

SCHEMBL61222

CC(C)(C)NC(=O)[C@H]1CC[C@H]2[C@@H]3CC=C4C=C(C(=O)O)CC[C@]4(C)[C@H]3CC[C@]12C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 15/20 1.00
SRD5A1 P18405 5/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Epristeride SCHEMBL23833504 1.00 SRD5A2 (1.00) SRD5A2SRD5A1
Epristeride SCHEMBL16115063 1.00 SRD5A2 (1.00) SRD5A2SRD5A1
Epristeride SCHEMBL5444493 1.00 SRD5A2 (1.00) SRD5A2SRD5A1
Epristeride SCHEMBL9782857 0.99 SRD5A2 (0.98) SRD5A2SRD5A1
SCHEMBL9114229 0.93 SRD5A2 (0.86) SRD5A2SRD5A1
SCHEMBL8994092 0.91 SRD5A2 (0.83) SRD5A2SRD5A1
SCHEMBL8151553 0.91 SRD5A2 (0.83) SRD5A2SRD5A1
SCHEMBL8151554 0.91 SRD5A2 (0.83) SRD5A2SRD5A1
Epristeride SCHEMBL9782855 0.91 SRD5A2 (0.83) SRD5A2SRD5A1
SCHEMBL9391082 0.90 SRD5A2 (0.82) SRD5A2SRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 10419 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260116861-A1 ISOXAZOLE HYDROXAMIC ACIDS AS HISTONE DEACETYLASE 6 INHIBITORS THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-04-30 US claimed
EP-4698175-A1 LYSINE ACETYLTRANSFERASE 6A (KAT6A) INHIBITOR, COMBINATIONS AND USES THEREOF Insilico Medicine IP Limited (HK) 2026-02-25 EP claimed
US-12522572-B2 Isoxazole hydroxamic acids as histone deacetylase 6 inhibitors THE GEORGE WASHINGTON UNIVERSITY, A CONGRESSIONALLY CHARTERED NOT-FOR-PROFIT CORPORATION (US) 2026-01-13 US claimed
US-20250295634-A1 USE OF ANTIANDROGENS TO TREAT SEPSIS RHODE ISLAND HOSPITAL 2025-09-25 US claimed
US-20250281509-A1 SEQUENTIAL HORMONE THERAPY TO IMPROVE SURVIVAL AND ENHANCE RESPONSE TO IMMUNE THERAPY IN MEN WITH PROSTATE CANCER THE JOHNS HOPKINS UNIVERSTY 2025-09-11 US claimed
EP-4608405-A1 COMPOSITIONS AND METHODS OF USE FOR MODIFIED RELEASE MINOXIDIL Veradermics, Incorporated (US) 2025-09-03 EP claimed
US-20250262192-A1 PROGNOSTIC PATHWAYS FOR HIGH RISK SEPSIS PATIENTS KONINKLIJKE PHILIPS N.V. (NL) 2025-08-21 US claimed
US-20250075180-A1 METHOD FOR EXPANSION CULTURE OF GAMMA-DELTA T CELL IMMUNOMAX CO., LTD. (KR) 2025-03-06 US claimed
EP-4499222-A2 COMPOSITIONS AND METHODS FOR PROMOTING HAIR GROWTH Locus Solutions IPCO, LLC (US) 2025-02-05 EP claimed
CN-119320422-A Eplerite impurity 17 beta- (N-tertiary butyl-amino-formyl) androstane-3, 5-diene-3-diphenyl phosphine oxide and preparation method and application thereof 江苏联环药业股份有限公司 2025-01-17 CN claimed
WO-1995006461-A1 STABILIZED TABLET FORMULATION SMITHKLINE BEECHAM CORPORATION (US) 1995-03-09 WO claimed
EP-0633892-A1 N-T-BUTYL-ANDROST-3,5-DIENE-17$g(b)-CARBOXAMIDE-3-CARBOXYLIC ACID POLYMORPH A SMITHKLINE BEECHAM CORPORATION (US) 1995-01-18 EP claimed
EP-0633781-A1 COMPOSITIONS AND METHODS FOR TREATING BENIGN PROSTATIC HYPERTROPHY SMITHKLINE BEECHAM CORPORATION (US) 1995-01-18 EP claimed
WO-1994017663-A1 TREATING ALOPECIA BY ADMINISTERING 5-ALPHA-REDUCTASE INHIBITING COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 1994-08-18 WO claimed
WO-1993019758-A1 COMPOSITIONS AND METHODS FOR TREATING BENIGN PROSTATIC HYPERTROPHY SMITHKLINE BEECHAM CORPORATION (US) 1993-10-14 WO claimed
WO-1993019080-A1 N-T-BUTYL-ANDROST-3,5-DIENE-17β-CARBOXAMIDE-3-CARBOXYLIC ACID POLYMORPH B SMITHKLINE BEECHAM CORPORATION (US) 1993-09-30 WO claimed
WO-1993019081-A1 N-T-BUTYL-ANDROST-3,5-DIENE-17β-CARBOXAMIDE-3-CARBOXYLIC ACID POLYMORPH A SMITHKLINE BEECHAM CORPORATION (US) 1993-09-30 WO claimed
EP-0289327-B1 STEROID 5-ALPHA-REDUCTASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1991-12-18 EP claimed
US-5017568-A Enzyme inhibitors, carboxylation SMITHKLINE BEECHAM CORPORATION (US) 1991-05-21 US claimed
EP-0289327-A2 Steroid 5-alpha-reductase inhibitors SMITHKLINE BEECHAM CORPORATION (US) 1988-11-02 EP claimed