Oenin

Oenin

SCHEMBL6139047

COc1cc(-c2[o+]c3cc(O)cc(O)c3cc2O[C@@H]2O[C@H](CO)[C@@H](O)[C@H](O)[C@H]2O)cc(OC)c1O

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CD38 P28907 3/20 0.74
DPP4 P27487 2/20 0.74
F2 P00734 1/20 0.66
MAOA P21397 1/20 0.56
TYR P14679 1/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
SLC28A3 Q9HAS3 2/20 0.49
ALDH1A1 P00352 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA13 Q8N1Q1 1/20 0.48
EPHX2 P34913 2/20 0.47
ACHE P22303 1/20 0.46
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oenin SCHEMBL676018 1.00 CD38 (0.74) CD38DPP4F2MAOATYR
Oenin SCHEMBL29894980 1.00 CD38 (0.74) CD38DPP4F2MAOATYR
Oenin SCHEMBL29468973 1.00 CD38 (0.74) CD38DPP4F2MAOATYR
Oenin SCHEMBL662772 1.00 CD38 (0.74) CD38DPP4F2MAOATYR
Oenin SCHEMBL29521448 1.00 CD38 (0.74) CD38DPP4F2MAOATYR
Oenin SCHEMBL723403 0.99 CD38 (0.73) CD38DPP4F2MAOATYR
Oenin SCHEMBL29881103 0.99 CD38 (0.73) CD38DPP4F2MAOATYR
Oenin SCHEMBL1096836 0.99 CD38 (0.73) CD38DPP4F2MAOATYR
SCHEMBL676805 0.99 CD38 (0.72) CD38DPP4F2MAOATYR
SCHEMBL30901362 0.98 CD38 (0.75) CD38DPP4F2MAOATYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1443948-B1 PROCESS FOR THE PREPARATION OF ANTHOCYANIN-CONTAINING PRODUCTS MEDPALETT PHARMACEUTICALS AS (NO) 2005-06-29 EP claimed
WO-2004096240-A1 ANTHOCYANINS USEFUL FOR THE TREATMENT OF DIABETES, CARDIOVASCULAR DISORDERS AND TO LOWER THE RISK OF ADVERSE EFFECTS OF HORMONE REPLACEMENT THERAPY MEDPALETT PHARMACEUTICALS AS (NO) 2004-11-11 WO claimed
EP-1443948-A1 PROCESS FOR THE PREPARATION OF ANTHOCYANIN-CONTAINING PRODUCTS Medpalett Pharmaceuticals AS (NO) 2004-08-11 EP claimed
US-20030091660-A1 Product MEDPALETT PHARMACEUTICALS AS (NO) 2003-05-15 US claimed
WO-2003039569-A1 PROCESS FOR THE PREPARATION OF ANTHOCYANIN-CONTAINAING PRODUCTS MEDPALETT PHARMACEUTICALS AS (NO) 2003-05-15 WO claimed
EP-1871402-B1 GRAPE CELL CULTURE FOR TREATING INFLAMMATION STATE OF ISRAEL MINI OF AGRICULTURE & RURAL DEV AGRICULTURAL RES ORGANIZATION (A R O ) VOLCANI CENTE (IL) 2017-07-26 EP disclosed
US-9308231-B2 Anti-inflammatory composition comprising malvidin-3-O-β-glucoside and a propolis extract Universite de Bordeaux (FR) 2016-04-12 US disclosed
US-6967032-B2 Mixtures of anthracyanins, monosaccharides, disaccharides MEDPALETT PHARMACEUTICALS AS (NO) 2005-11-22 US disclosed
EP-1443948-B1 PROCESS FOR THE PREPARATION OF ANTHOCYANIN-CONTAINING PRODUCTS MEDPALETT PHARMACEUTICALS AS (NO) 2005-06-29 EP disclosed
WO-2005009140-A1 USE OF ANTHOCYANINS IN FISH FOOD BIOCHEM LABORATORIES AS (NO) 2005-02-03 WO disclosed
EP-1443948-A1 PROCESS FOR THE PREPARATION OF ANTHOCYANIN-CONTAINING PRODUCTS Medpalett Pharmaceuticals AS (NO) 2004-08-11 EP disclosed
US-20030091660-A1 Product MEDPALETT PHARMACEUTICALS AS (NO) 2003-05-15 US disclosed
WO-2003039569-A1 PROCESS FOR THE PREPARATION OF ANTHOCYANIN-CONTAINAING PRODUCTS MEDPALETT PHARMACEUTICALS AS (NO) 2003-05-15 WO disclosed
WO-1998038316-A1 BETA-GLUCOSIDASES, METHODS FOR OBTAINING SAME, PREPARATIONS CONTAINING SAID BETA-GLUCOSIDASES AND USES THEREOF DSM N.V. (NL) 1998-09-03 WO disclosed