SCHEMBL6140002

SCHEMBL6140002

O=C(NC(Cc1ccc2nc(-c3c(F)cccc3Cl)ccc2c1)C(=O)O)c1c(Cl)cccc1Cl

nearest known ligand 0.87

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 17/20 0.87
ITGAV P06756 4/20 0.87
ITGA4 P13612 11/20 0.61
ITGB7 P26010 5/20 0.61
ITGA5 P08648 5/20 0.50
ITGB3 P05106 2/20 0.50
ITGB2 P05107 2/20 0.48
ICAM1 P05362 2/20 0.48
ITGAL P20701 2/20 0.48
ITGA2 P17301 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3314255 1.00 ITGB1 (0.87) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3315902 0.97 ITGB1 (0.85) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3315359 0.96 ITGB1 (0.80) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL6139776 0.94 ITGB1 (0.77) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3313255 0.94 ITGB1 (0.77) ITGB1ITGAVITGA4ITGB7ITGA2
SCHEMBL3316690 0.93 ITGB1 (0.85) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3313373 0.93 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL8352229 0.93 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3316398 0.93 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7ITGA5
SCHEMBL3313356 0.93 ITGB1 (1.00) ITGB1ITGAVITGA4ITGB7ITGA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed