SCHEMBL6140359

SCHEMBL6140359

Cc1ccc(S(=O)(=O)[C@H]2CCCCN2C(=O)NC(Cc2ccc3nc(-c4c(Cl)cccc4Cl)ccc3c2)C(=O)O)cc1

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.55
ITGAV P06756 1/20 0.55
ITGA4 P13612 13/20 0.43
ITGB7 P26010 5/20 0.43
ALDH1A1 P00352 2/20 0.42
HSD17B10 Q99714 1/20 0.42
KCNH2 Q12809 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6140351 0.94 ITGB1 (0.48) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL6140062 0.92 ITGB1 (0.59) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL6139884 0.90 ITGB1 (0.59) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL6142066 0.88 ITGB1 (0.45) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL6140246 0.87 ITGB1 (0.51) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL6141601 0.86 ITGB1 (0.39) ITGB1ITGAVITGA4ALDH1A1HSD17B10
SCHEMBL3320849 0.84 ITGB1 (0.56) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL3317244 0.80 ITGB1 (0.70) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL4410500 0.79 ITGB1 (0.53) ITGB1ITGAVITGA4ITGB7ALDH1A1
SCHEMBL3317863 0.79 ITGB1 (0.53) ITGB1ITGAVITGA4ITGB7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed