SCHEMBL6142209

SCHEMBL6142209

[O]c1ccc(-c2cccnc2)cc1Cl

nearest known ligand 0.65

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 6/20 0.65
MKNK2 Q9HBH9 6/20 0.65
CYP2A6 P11509 3/20 0.54
CYP1A2 P05177 2/20 0.54
ALDH1A1 P00352 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP11B1 P15538 5/20 0.51
CYP11B2 P19099 5/20 0.51
CYP19A1 P11511 3/20 0.51
CYP17A1 P05093 1/20 0.51
MEN1 O00255 1/20 0.49
PSIP1 O75475 1/20 0.49
AXL P30530 1/20 0.49
KDR P35968 1/20 0.48
ERN1 O75460 1/20 0.47
KMO O15229 1/20 0.47
NPY5R Q15761 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27636086 0.79 ESR2 (0.61) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL12491570 0.79 MKNK1 (0.60) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL30137140 0.79 ESR2 (0.61) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL13890275 0.78 MKNK1 (0.56) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL14715531 0.77 ESR2 (0.57) CYP2A6CYP1A2ALDH1A1MEN1
SCHEMBL21753332 0.76 MKNK1 (0.54) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL25463021 0.75 CYP11B1 (0.56) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL21770157 0.75 MKNK1 (0.56) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL12103445 0.74 CYP2A6 (0.79) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1
SCHEMBL17951830 0.74 CYP2A6 (0.79) MKNK1MKNK2CYP2A6CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1558567-A1 NOVEL AMIDE COMPOUNDS WITH MCH ANTAGONISTIC EFFECT AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2005-08-03 EP disclosed
WO-2004039764-A1 NOVEL AMIDE COMPOUNDS WITH MCH ANTAGONISTIC EFFECT AND MEDICAMENTS COMPRISING SAID COMPOUNDS BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-05-13 WO disclosed