SCHEMBL6146929

SCHEMBL6146929

CS(=O)(=O)c1ccc(-c2c(Oc3ccc(OCCC4CCCCN4)cc3)ccc3cc(O)ccc23)cc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 13/20 0.51
ESR2 Q92731 12/20 0.51
CHEK2 O96017 1/20 0.41
SSTR2 P30874 1/20 0.39
LTA4H P09960 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6148234 0.87 ESR1 (0.69) ESR1ESR2CHEK2SSTR2
Hydrochloric Acid SCHEMBL6111606 0.86 ESR1 (0.69) ESR1ESR2CHEK2SSTR2
Hydrochloric Acid SCHEMBL6231092 0.82 ESR1 (0.53) ESR1ESR2CHEK2SSTR2
Hydrochloric Acid SCHEMBL6234142 0.82 ESR1 (0.70) ESR1ESR2CHEK2SSTR2LTA4H
SCHEMBL6232447 0.80 ESR1 (0.57) ESR1ESR2SSTR2
SCHEMBL6232806 0.80 ESR1 (0.57) ESR1ESR2CHEK2SSTR2
SCHEMBL6234735 0.80 ESR1 (0.69) ESR1ESR2CHEK2SSTR2
Hydrochloric Acid SCHEMBL6230778 0.79 ESR1 (0.68) ESR1ESR2
SCHEMBL6238234 0.78 ESR1 (0.53) ESR1ESR2CHEK2SSTR2
SCHEMBL6239106 0.78 ESR1 (0.45) ESR1ESR2CHEK2SSTR2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1601356-A1 CRYSTALLINE NON-SOLVATED 1-(4-(2-PIPERIDINYLETHOXY)PHENOXY)-2-(4-METHANESULFONYLPHENYL)-6-HYDROXYNAPHTHALENE HYDROCHLORIDE Eli Lilly and Company (US) 2005-12-07 EP disclosed
WO-2004075894-A1 CRYSTALLINE NON-SOLVATED 1-(4-(2-PIPERIDINYLETHOXY)PHENOXY)-2-(4-METHANESULFONYLPHENYL)-6-HYDROXYNAPHTHALENE HYDROCHLORIDE ELI LILLY AND COMPANY (US) 2004-09-10 WO disclosed