SCHEMBL6147350

SCHEMBL6147350

CCNC(=O)ON1CC2CN(CCCC(Oc3ccc(OC)c(OC)c3)c3ccc(C#N)cc3)CC(C1)O2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.39
SLC6A4 P31645 2/20 0.37
HRH3 Q9Y5N1 1/20 0.37
DRD3 P35462 3/20 0.36
MCHR1 Q99705 1/20 0.35
MGLL Q99685 2/20 0.33
KEAP1 Q14145 2/20 0.33
NFE2L2 Q16236 2/20 0.33
HIF1A Q16665 1/20 0.33
SLC6A2 P23975 2/20 0.33
TMEM97 Q5BJF2 1/20 0.33
CYP2D6 P10635 1/20 0.33
NOS2 P35228 1/20 0.33
ADRA1D P25100 2/20 0.32
ADRA1A P35348 2/20 0.32
ADRA1B P35368 2/20 0.32
CACNA1F O60840 1/20 0.32
HTR1A P08908 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
DRD2 P14416 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2964357 0.89 POLB (0.39) KCNH2SLC6A4HRH3DRD3MCHR1
SCHEMBL2966856 0.85 SLC6A4 (0.40) KCNH2SLC6A4HRH3DRD3MCHR1
SCHEMBL2966873 0.84 KCNH2 (0.39) KCNH2SLC6A4HRH3DRD3MCHR1
SCHEMBL2968077 0.84 HRH3 (0.42) KCNH2SLC6A4HRH3DRD3MCHR1
SCHEMBL2964346 0.82 MCHR1 (0.43) KCNH2SLC6A4HRH3MCHR1TMEM97
SCHEMBL6095424 0.82 POLB (0.41) SLC6A4HRH3DRD3MCHR1HIF1A
SCHEMBL2959501 0.81 KCNH2 (0.38) KCNH2SLC6A4HRH3DRD3MCHR1
SCHEMBL4414313 0.81 PDE4B (0.39) KCNH2SLC6A4HRH3MAPT
SCHEMBL5965486 0.81 MCHR1 (0.40) SLC6A4HRH3DRD3MCHR1KEAP1
SCHEMBL6739004 0.81 POLB (0.40) SLC6A4HRH3DRD3MCHR1HIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235831-B1 NEW OXABISPIDINE COMPOUNDS USEFUL IN THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2005-03-30 EP claimed