SCHEMBL61480

SCHEMBL61480

CCc1cccc(CC)c1-c1nc(C)c(CN(C)[C@H]2CCCc3ccccc32)c(N2CCN(C(CC)C(=O)O)CC2)n1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
P4HB P07237 1/20 0.38
CXCR4 P61073 5/20 0.35
ALDH1A1 P00352 1/20 0.35
XBP1 P17861 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.34
TMEM97 Q5BJF2 3/20 0.33
SIGMAR1 Q99720 2/20 0.33
P2RX3 P56373 2/20 0.33
P2RX2 Q9UBL9 2/20 0.33
KCNH2 Q12809 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL63771 0.90 CXCR4 (0.38) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL62217 0.88 MEN1 (0.40) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL63372 0.88 CXCR4 (0.42) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL63341 0.88 CXCR4 (0.44) MEN1KMT2AP4HBCXCR4KCNH2
SCHEMBL62216 0.88 MEN1 (0.40) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL62204 0.88 MEN1 (0.40) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL62583 0.87 MEN1 (0.43) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL72863 0.87 MEN1 (0.42) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL62909 0.87 MEN1 (0.42) MEN1KMT2AP4HBCXCR4ALDH1A1
SCHEMBL61753 0.87 MEN1 (0.40) MEN1KMT2AP4HBCXCR4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8129395-B2 4,5-disubstituted-2-aryl pyrimidines NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-03-06 US disclosed