SCHEMBL6150797

SCHEMBL6150797

COC(=O)[C@H](Cc1ccc(OC(=O)N(C)C)cc1)NC(=O)C12CC3CC(C1)CC(C(=O)OC)(C3)C2

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.59
KMT2A Q03164 2/20 0.59
ALDH1A1 P00352 2/20 0.43
ITGB1 P05556 4/20 0.43
ITGA4 P13612 4/20 0.43
MAPT P10636 3/20 0.41
CYP2D6 P10635 1/20 0.41
KLKB1 P03952 1/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 3/20 0.38
ABL1 P00519 1/20 0.38
RIN1 Q13671 1/20 0.38
CYP3A4 P08684 2/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5859743 0.94 KMT2A (0.51) NPSR1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL5860871 0.92 KMT2A (0.48) NPSR1KMT2AITGB1ITGA4MAPT
SCHEMBL5861047 0.92 KMT2A (0.59) NPSR1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL5862666 0.92 KMT2A (0.49) NPSR1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL5859893 0.87 KMT2A (0.60) NPSR1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL6150500 0.87 KMT2A (0.55) NPSR1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL5859997 0.85 KMT2A (0.64) NPSR1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL5861027 0.84 KMT2A (0.47) NPSR1KMT2AITGB1ITGA4MAPT
SCHEMBL5859608 0.84 KMT2A (0.48) NPSR1KMT2AALDH1A1ITGB1ITGA4
SCHEMBL5862652 0.84 KMT2A (0.44) NPSR1KMT2AITGB1ITGA4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1144364-B1 MULTICYCLIC COMPOUNDS WHICH INHIBIT LEUKOCYTE ADHESION MEDIATED BY VLA-4 ELAN PHARM INC (US) 2005-07-13 EP claimed