SCHEMBL6151547

SCHEMBL6151547

Cc1ccc(C=CCc2sccc2S(=O)(=O)Nc2onc(C)c2Br)c(C)c1

nearest known ligand 0.75

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
EDNRB P24530 20/20 0.75
EDNRA P25101 20/20 0.75

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6151545 1.00 EDNRB (0.75) EDNRBEDNRA
SCHEMBL4631568 0.87 EDNRA (0.73) EDNRBEDNRA
SCHEMBL4631567 0.87 EDNRA (0.73) EDNRBEDNRA
SCHEMBL4632359 0.86 EDNRB (0.79) EDNRBEDNRA
SCHEMBL4632361 0.86 EDNRB (0.79) EDNRBEDNRA
SCHEMBL4630707 0.86 EDNRB (0.77) EDNRBEDNRA
SCHEMBL4630702 0.86 EDNRB (0.77) EDNRBEDNRA
SCHEMBL6151669 0.82 EDNRB (1.00) EDNRBEDNRA
SCHEMBL6151714 0.80 EDNRB (1.00) EDNRBEDNRA
SCHEMBL4632393 0.80 EDNRA (1.00) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5962490-A Thienyl-, furyl- and pyrrolyl-sulfonamides and derivatives thereof that modulate the activity of endothelin TEXAS BIOTECHNOLOGY CORPORATION (US) 1999-10-05 US claimed
CN-1636994-B Process of preparing alkali metal salys of hydrophobic sulfonamides and alkali metal salt produced thereby ENCYSIVE PHARMACEUTICALS INC 2010-05-12 CN disclosed
CN-100558724-C Adjust active sulphonamide of endothelium peptide and derivative thereof ANSEHIV PHARMACEUTICAL CORP (US) 2009-11-11 CN disclosed
CN-1215069-C Sulfonamides and derivatives thereof that modulate the activity of endothelin ENCYSIVE PHARMACEUTICALS INC (US) 2005-08-17 CN disclosed
CN-1636994-A Process of preparing alkali metal salys of hydrophobic sulfonamides and alkali metal salt produced thereby ENCYSIVE PHARMACEUTICALS INC (US) 2005-07-13 CN disclosed
EP-0980369-B1 SULFONAMIDES FOR TREATMENT OF ENDOTHELIN-MEDIATED DISORDERS ENCYSIVE PHARMACEUTICALS INC (US) 2005-03-30 EP disclosed
EP-1498419-A1 Process for preparing alkali metal salts of hydrophobic sulfonamides ENCYSIVE PHARMACEUTICALS INC. (US) 2005-01-19 EP disclosed
EP-1498418-A1 Sulfonamides for treatment of endothelin-mediated disorders ENCYSIVE PHARMACEUTICALS INC. (US) 2005-01-19 EP disclosed
CN-1179961-C Sulfonamides for the treatment of endothelin mediated diseases ��ɪϣ����ҩ��˾ 2004-12-15 CN disclosed
CN-1530366-A Sulphonic acid amide for regulating bast peptide activity and derivative thereof ��ɪϣ����ҩ��˾ 2004-09-22 CN disclosed
EP-0946552-B1 SULFONAMIDES AND DERIVATIVES THEREOF THAT MODULATE THE ACTIVITY OF ENDOTHELIN ENCYSIVE PHARMACEUTICALS INC (US) 2004-07-07 EP disclosed
CN-1253560-A Sulfonamides for the treatment of endothelin mediated diseases TEXA BIOTECHNOLOGY CORP (US) 2000-05-17 CN disclosed
CN-1231664-A Sulfonamides and derivatives thereof that modulate the activity of endothelin TEXAS BIOTECHNOLOGY CORP (US) 1999-10-13 CN disclosed