SCHEMBL6152154

SCHEMBL6152154

CCCCC1CCc2c(cc(F)c(OC)c2Cl)C1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 6/20 0.32
DRD2 P14416 5/20 0.32
CYP3A4 P08684 2/20 0.32
CYP2C8 P10632 2/20 0.32
S1PR3 Q99500 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
SGPL1 O95470 1/20 0.32
HTR1A P08908 1/20 0.31
DRD4 P21917 1/20 0.31
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
DPP4 P27487 2/20 0.30
SMYD3 Q9H7B4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4853543 0.74 CYP24A1 (0.33) DRD3DRD2SGPL1HTR1ADRD4
SCHEMBL2419510 0.71 MEN1 (0.31)
SCHEMBL5722716 0.70 CYP3A4 (0.42) DRD3DRD2CYP3A4CYP2C8S1PR3
SCHEMBL7793664 0.70 CYP3A4 (0.42) DRD3DRD2CYP3A4CYP2C8S1PR3
SCHEMBL31545566 0.69 CYP3A4 (0.42) DRD3DRD2CYP3A4CYP2C8S1PR3
SCHEMBL24225295 0.69 ACACB (0.35)
SCHEMBL7792870 0.68 CYP3A4 (0.40) DRD3DRD2CYP3A4CYP2C8S1PR3
SCHEMBL7793326 0.68 CYP3A4 (0.40) DRD3DRD2CYP3A4CYP2C8S1PR3
SCHEMBL10893945 0.67 CYP1A2 (0.37) CYP2D6CYP2C9CYP2C19DPP4
SCHEMBL10893934 0.67 CYP1A2 (0.37) CYP2D6CYP2C9CYP2C19DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551820-A2 ESTROGEN RECEPTOR MODULATORS Merck & Co., Inc. (US) 2005-07-13 EP disclosed
WO-2004026887-A2 ESTROGEN RECEPTOR MODULATORS MERCK & CO., INC. (US) 2004-04-01 WO disclosed