SCHEMBL6152269

SCHEMBL6152269

CN(C)CC(=O)NCC1CCN(C(=O)CCC(NC(=O)[C@@H]2CCCN2S(=O)(=O)c2cc(Cl)cc(Cl)c2)C(=O)O)CC1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 18/20 0.51
ITGA4 P13612 17/20 0.51
ITGB7 P26010 3/20 0.46
ITGA2 P17301 1/20 0.43
ITGAV P06756 1/20 0.41
ITGA5 P08648 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6401872 1.00 ITGB1 (0.51) ITGB1ITGA4ITGB7ITGA2ITGAV
SCHEMBL6147979 1.00 ITGB1 (0.51) ITGB1ITGA4ITGB7ITGA2ITGAV
SCHEMBL6158932 0.92 ITGB1 (0.46) ITGB1ITGA4ITGB7
SCHEMBL6158937 0.92 ITGB1 (0.46) ITGB1ITGA4ITGB7
SCHEMBL6401850 0.91 ITGB1 (0.53) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6401858 0.91 ITGB1 (0.53) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6401876 0.89 ITGB1 (0.57) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6401871 0.89 ITGB1 (0.57) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6156368 0.88 ITGB1 (0.51) ITGB1ITGA4ITGB7ITGA2
SCHEMBL6156360 0.88 ITGB1 (0.51) ITGB1ITGA4ITGB7ITGA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495044-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. Uriach y Compania S.A. (ES) 2005-01-12 EP disclosed
WO-2003084984-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. URIACH Y COMPANIA S.A. (ES) 2003-10-16 WO disclosed