SCHEMBL6152647

SCHEMBL6152647

CC(C)n1cnc2c(NCc3ccc(Cl)cc3)nc(Cl)nc21

nearest known ligand 0.82

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 7/20 0.82
CDK5 Q00535 8/20 0.69
CDK5R1 Q15078 6/20 0.69
CDK2 P24941 5/20 0.67
CCNE1 P24864 4/20 0.67
CCNE2 O96020 3/20 0.64
TDP1 Q9NUW8 2/20 0.63
KDM4E B2RXH2 2/20 0.63
NPC1 O15118 2/20 0.63
MAPT P10636 2/20 0.63
CCNB2 O95067 1/20 0.63
CCNB1 P14635 1/20 0.63
CCNB3 Q8WWL7 1/20 0.63
CCNA2 P20248 2/20 0.61
CCNA1 P78396 2/20 0.61
DYRK1A Q13627 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28771322 0.91 CDK1 (0.79) CDK1CDK5CDK5R1CDK2CCNE1
SCHEMBL31072401 0.91 CDK1 (0.79) CDK1CDK5CDK5R1CDK2CCNE1
SCHEMBL28459824 0.91 CDK1 (0.79) CDK1CDK5CDK5R1CDK2CCNE1
SCHEMBL1400442 0.90 CDK1 (1.00) CDK1CDK5CDK2CCNE1TDP1
SCHEMBL1443236 0.89 TDP1 (0.80) CDK1CDK5CDK5R1CDK2CCNE1
SCHEMBL17628615 0.89 CDK1 (0.87) CDK1CDK5CDK2CCNE1CCNE2
SCHEMBL27581376 0.88 CDK5 (0.66) CDK1CDK5CDK5R1CDK2CCNE1
SCHEMBL28461058 0.88 CDK1 (0.78) CDK1CDK5CDK5R1CDK2CCNE1
SCHEMBL1443449 0.87 CDK1 (0.73) CDK1CDK5CDK5R1CDK2CCNE1
SCHEMBL6821050 0.86 CDK1 (0.79) CDK1CDK5CDK2TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1150982-B1 PURINE INHIBITORS OF CYCLIN DEPENDENT KINASE 2 AND IkB-alpha CV THERAPEUTICS INC (US) 2005-10-12 EP disclosed