SCHEMBL6156903

SCHEMBL6156903

CCCCCCCNC(=O)N(C)c1cccc(-c2ccc(CC(Nc3ccccc3C(=O)c3ccccc3)C(=O)N3CCN(C(=O)O)C(C(C)(C)C)C3)cc2)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 17/20 0.36
PTPN1 P18031 1/20 0.34
PPARA Q07869 2/20 0.33
HPN P05981 1/20 0.33
ST14 Q9Y5Y6 1/20 0.33
TACR1 P25103 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2849746 1.00 PPARG (0.36) PPARGPTPN1PPARAHPNST14
SCHEMBL2851730 0.90 PPARG (0.41) PPARGPPARAHPNST14
SCHEMBL2851732 0.90 PPARG (0.41) PPARGPPARAHPNST14
SCHEMBL2859244 0.87 PPARG (0.40) PPARGPPARAHPNST14
SCHEMBL2859247 0.87 PPARG (0.40) PPARGPPARAHPNST14
SCHEMBL2849743 0.86 PPARG (0.46) PPARGPTPN1
SCHEMBL2854526 0.86 PPARG (0.40) PPARGPPARA
SCHEMBL2854528 0.86 PPARG (0.40) PPARGPPARA
SCHEMBL2851721 0.85 PPARG (0.39) PPARGPPARA
SCHEMBL2851713 0.85 PPARG (0.39) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575911-A2 BIAROMATIC COMPOUNDS WHICH ACTIVATE PPAR-GAMMA TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS Galderma Research & Development, S.N.C. (FR) 2005-09-21 EP disclosed
WO-2004046091-A2 BIAROMATIC COMPOUNDS WHICH ACTIVATE PPAR-GAMA TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-06-03 WO disclosed