SCHEMBL6156934

SCHEMBL6156934

COC(=O)C(Cc1ccc2nc(-c3c(Cl)cccc3Cl)ccc2c1)N(C(=O)Nc1c(Cl)cccc1Cl)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 4/20 0.51
ITGAV P06756 1/20 0.51
ABL1 P00519 1/20 0.37
ITGA4 P13612 3/20 0.33
ITGB7 P26010 2/20 0.33
CDK2 P24941 1/20 0.33
TACR3 P29371 2/20 0.33
SCN9A Q15858 1/20 0.33
LCK P06239 1/20 0.33
KCNH2 Q12809 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CTNNB1 P35222 1/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
HPGD P15428 2/20 0.32
DGAT1 O75907 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4624847 0.81 ITGB1 (0.55) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL3314709 0.79 ITGB1 (0.63) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL3312626 0.79 ITGB1 (0.53) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL3321001 0.78 ITGB1 (0.60) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL6146195 0.78 ITGB1 (0.54) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL5127858 0.78 ITGB1 (0.71) ITGB1ITGAVITGA4ITGB7
SCHEMBL3313415 0.77 ITGB1 (0.59) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL4750010 0.77 ITGB1 (0.59) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL13398404 0.77 ITGB1 (0.64) ITGB1ITGAVABL1ITGA4ITGB7
SCHEMBL3316824 0.74 ITGB1 (0.56) ITGB1ITGAVABL1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406932-A4 QUICK CURING COMPOSITION KANEKA CORP (JP) 2005-03-23 EP disclosed
EP-1501801-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2005-02-02 EP disclosed
EP-1406932-A1 QUICK CURING COMPOSITION KANEKA CORPORATION (JP) 2004-04-14 EP disclosed
WO-2003093237-A1 2,6-QUINOLINYL AND 2,6-NAPHTHYL DERIVATIVES, PROCESSES FOR PREPARING THEM AND THEIR USES AS VLA-4 INHIBITORS UCB, S.A. (BE) 2003-11-13 WO disclosed
WO-2003000749-A1 QUICK CURING COMPOSITION KANEKA CORPORATION (JP) 2003-01-03 WO disclosed