SCHEMBL6157260

SCHEMBL6157260

COC(=O)C(CCC(=O)N1CCC(CNC(=O)N2CCN(C)CC2)CC1)NC(=O)[C@H]1CCCN1S(=O)(=O)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 14/20 0.45
ITGA4 P13612 14/20 0.45
ITGB7 P26010 1/20 0.41
CCKBR P32239 4/20 0.41
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
CASP1 P29466 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6157254 1.00 ITGB1 (0.45) ITGB1ITGA4ITGB7CCKBRHCRTR1
SCHEMBL6155691 0.93 ITGB1 (0.50) ITGB1ITGA4ITGB7CCKBRCASP1
SCHEMBL6155700 0.93 ITGB1 (0.50) ITGB1ITGA4ITGB7CCKBRCASP1
SCHEMBL6151156 0.89 ITGB1 (0.46) ITGB1ITGA4ITGB7CCKBRHCRTR1
SCHEMBL6151159 0.89 ITGB1 (0.46) ITGB1ITGA4ITGB7CCKBRHCRTR1
SCHEMBL6158937 0.87 ITGB1 (0.46) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6158932 0.87 ITGB1 (0.46) ITGB1ITGA4ITGB7HCRTR1HCRTR2
SCHEMBL6156360 0.86 ITGB1 (0.51) ITGB1ITGA4ITGB7
SCHEMBL6156368 0.86 ITGB1 (0.51) ITGB1ITGA4ITGB7
SCHEMBL6401091 0.84 ITGB1 (0.48) ITGB1ITGA4ITGB7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1495044-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. Uriach y Compania S.A. (ES) 2005-01-12 EP disclosed
WO-2003084984-A1 HETEROCYCLIC AMIDES WITH ALPHA-4 INTEGRIN ANTAGONIST ACTIVITY J. URIACH Y COMPANIA S.A. (ES) 2003-10-16 WO disclosed