SCHEMBL6158824

SCHEMBL6158824

CC(=O)S[C@@H]1CC(=O)N(Cc2ccc(Oc3ccccc3)cc2)[C@H]1C

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 6/20 0.45
HCRTR2 O43614 6/20 0.45
SIGMAR1 Q99720 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
FAAH O00519 2/20 0.38
HRH3 Q9Y5N1 1/20 0.38
SRD5A2 P31213 1/20 0.38
LTA4H P09960 1/20 0.38
FFAR1 O14842 1/20 0.37
MGLL Q99685 1/20 0.37
ALDH1A1 P00352 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6159439 1.00 HCRTR1 (0.45) HCRTR1HCRTR2SIGMAR1MEN1KMT2A
SCHEMBL6157560 0.88 HCRTR1 (0.44) HCRTR1HCRTR2MEN1KMT2AFAAH
SCHEMBL6157562 0.88 HCRTR1 (0.44) HCRTR1HCRTR2MEN1KMT2AFAAH
SCHEMBL6157564 0.88 HCRTR1 (0.44) HCRTR1HCRTR2MEN1KMT2AFAAH
SCHEMBL6157486 0.87 HCRTR1 (0.44) HCRTR1HCRTR2MEN1KMT2AFAAH
SCHEMBL6157490 0.87 HCRTR1 (0.44) HCRTR1HCRTR2MEN1KMT2AFAAH
SCHEMBL6157488 0.87 HCRTR1 (0.44) HCRTR1HCRTR2MEN1KMT2AFAAH
SCHEMBL6157435 0.86 HCRTR1 (0.43) HCRTR1HCRTR2SIGMAR1MEN1KMT2A
SCHEMBL6157425 0.86 HCRTR1 (0.43) HCRTR1HCRTR2SIGMAR1MEN1KMT2A
SCHEMBL6158372 0.86 HCRTR1 (0.43) HCRTR1HCRTR2SIGMAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed