SCHEMBL6159525

SCHEMBL6159525

O=C1C[C@@H](SS[C@@H]2CC(=O)N(Cc3ccc(Oc4ccccc4)cc3)C2)CN1Cc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.49
TSHR P16473 1/20 0.49
HCRTR1 O43613 3/20 0.43
HCRTR2 O43614 3/20 0.43
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
DPP4 P27487 1/20 0.41
CNR2 P34972 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PTPN1 P18031 1/20 0.40
GRM2 Q14416 1/20 0.40
MMP2 P08253 1/20 0.40
EGLN1 Q9GZT9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6158330 1.00 HPGD (0.49) HPGDTSHRHCRTR1HCRTR2HTT
SCHEMBL6158326 1.00 HPGD (0.49) HPGDTSHRHCRTR1HCRTR2HTT
SCHEMBL6158859 0.90 HPGD (0.43) HPGDTSHRHCRTR1HCRTR2HTT
SCHEMBL6158788 0.90 HPGD (0.47) HPGDTSHRHCRTR1HCRTR2HTT
SCHEMBL6157836 0.89 TSHR (0.42) HPGDTSHRHCRTR1HCRTR2SMN1; SMN2
SCHEMBL6157901 0.87 HCRTR1 (0.44) HPGDTSHRHCRTR1HCRTR2CNR2
SCHEMBL6157459 0.86 SMN1; SMN2 (0.43) TSHRHCRTR1HCRTR2SMN1; SMN2KMT2A
SCHEMBL6160144 0.85 SMN1; SMN2 (0.45) HPGDTSHRHCRTR1HCRTR2HTT
SCHEMBL6158423 0.85 SMN1; SMN2 (0.45) HPGDTSHRHCRTR1HCRTR2HTT
SCHEMBL6157442 0.85 HCRTR1 (0.46) HPGDTSHRHCRTR1HCRTR2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed