SCHEMBL6159575

SCHEMBL6159575

O=C(O)CCNC(=O)SC1CCC(=O)N1Cc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 4/20 0.48
HCRTR2 O43614 4/20 0.48
FFAR1 O14842 1/20 0.41
EGLN1 Q9GZT9 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
SRD5A2 P31213 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
CHRM4 P08173 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.39
P2RX7 Q99572 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6158757 0.90 EGLN1 (0.49) HCRTR1HCRTR2EGLN1HDAC1HDAC6
SCHEMBL6159505 0.88 HDAC1 (0.51) HCRTR1HCRTR2HDAC1HDAC6HRH3
SCHEMBL6160370 0.85 HCRTR1 (0.51) HCRTR1HCRTR2FFAR1EGLN1HDAC1
SCHEMBL6158510 0.84 HCRTR1 (0.52) HCRTR1HCRTR2EGLN1HDAC1HDAC6
SCHEMBL6157202 0.83 HCRTR1 (0.53) HCRTR1HCRTR2FFAR1EGLN1HDAC1
SCHEMBL6158664 0.82 HCRTR1 (0.48) HCRTR1HCRTR2EGLN1HDAC1HDAC6
SCHEMBL6162062 0.82 HCRTR1 (0.56) HCRTR1HCRTR2HDAC1HDAC6
SCHEMBL6159092 0.81 HCRTR1 (0.51) HCRTR1HCRTR2FFAR1EGLN1HDAC1
SCHEMBL6159008 0.80 HCRTR1 (0.55) HCRTR1HCRTR2FFAR1EGLN1HDAC1
SCHEMBL6160316 0.80 HCRTR2 (0.53) HCRTR1HCRTR2HDAC1HDAC6ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953789-B2 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-10-11 US disclosed
US-6420415-B1 Thiol compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-07-16 US disclosed