SCHEMBL6163498

SCHEMBL6163498

CC1(C)CC(=O)c2cnn(-c3ccccc3)c2C1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA4 P22748 10/20 0.69
CA2 P00918 8/20 0.69
CA1 P00915 5/20 0.69
CA9 Q16790 1/20 0.68
ALDH1A1 P00352 5/20 0.60
KMT2A Q03164 3/20 0.60
MEN1 O00255 2/20 0.60
HPGD P15428 2/20 0.60
KDM4E B2RXH2 2/20 0.60
GFER P55789 1/20 0.60
HSD11B1 P28845 1/20 0.50
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.47
CYP11B2 P19099 1/20 0.45
HIF1A Q16665 1/20 0.44
LMNA P02545 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1220588 0.85 CA4 (0.65) CA4CA2CA1CA9ALDH1A1
SCHEMBL7536254 0.83 CA4 (0.66) CA4CA2CA1CA9ALDH1A1
SCHEMBL1220443 0.83 CA4 (0.65) CA4CA2CA1CA9ALDH1A1
SCHEMBL14980286 0.82 CA4 (0.65) CA4CA2CA1CA9ALDH1A1
SCHEMBL1219306 0.81 CA4 (0.67) CA4CA2CA1CA9ALDH1A1
SCHEMBL13828097 0.79 CA4 (0.61) CA4CA2CA1CA9ALDH1A1
SCHEMBL408184 0.79 CA4 (0.61) CA4CA2CA1CA9ALDH1A1
SCHEMBL21172119 0.79 CA4 (0.61) CA4CA2CA1CA9ALDH1A1
SCHEMBL13848537 0.78 CA4 (0.49) CA4CA2CA1CA9ALDH1A1
SCHEMBL19117746 0.76 CA4 (0.56) CA4CA2CA1CA9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-B1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-04-20 EP disclosed
US-6716856-B1 CELL PROLIFERATIVE DISORDERS OR ALZHEIMER'S DISEASE; REDUCED TOXICITY; CDK/CYCLIN KINASE INHIBITORY ACTIVITY PHARMACIA & TUBJOHN SPA (IT) 2004-04-06 US disclosed