SCHEMBL6166675

SCHEMBL6166675

CC(C)(C)[C@@]1(C#N)CCCN1C(=O)CN

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 6/20 0.38
DPP8 Q6V1X1 1/20 0.32
DPP9 Q86TI2 1/20 0.32
CTSS P25774 4/20 0.32
CTSK P43235 4/20 0.32
CTSB P07858 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1150768 0.82 DPP4 (0.35) DPP4DPP8DPP9
SCHEMBL3186817 0.82 DPP4 (0.35) DPP4DPP8DPP9
SCHEMBL23247420 0.78 DPP4 (0.32) DPP4DPP8DPP9CTSSCTSK
SCHEMBL82542 0.78 DPP4 (0.32) DPP4DPP8DPP9CTSSCTSK
SCHEMBL22964983 0.71 DPP4 (0.35) DPP4DPP8DPP9
SCHEMBL6169498 0.70 MAPT (0.43) DPP4DPP8DPP9CTSS
SCHEMBL4660548 0.69 DPP4 (0.40) DPP4DPP8DPP9
SCHEMBL6166415 0.69 MAPT (0.42) DPP4DPP8DPP9CTSS
SCHEMBL3959337 0.67 DPP4 (0.33) DPP4DPP8DPP9
SCHEMBL28523847 0.67 DPP4 (0.33) DPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1465891-A4 INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARM INC (US) 2005-08-17 EP disclosed
US-20050070719-A1 Inhibitors of dipeptidyl peptidase iv GUILFORD PHARMACEUTICALS 2005-03-31 US disclosed
EP-1465891-A2 INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS INC. (US) 2004-10-13 EP disclosed
WO-2003057666-A2 INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS (US) 2003-07-17 WO disclosed
WO-2003057144-A2 CHANGE INHIBITORS OF DIPEPTIDYL PEPTIDASE IV GUILFORD PHARMACEUTICALS (US) 2003-07-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050070719-A1 Inhibitors of dipeptidyl peptidase iv DPP4, DPP3, DPP7 DPP4 1/4885DPP8 5/4885DPP9 4/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.