SCHEMBL6168868

SCHEMBL6168868

CCOC(=O)c1cn(Cc2cccc(C=NN)c2)cc1-c1ccc(-c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 6/20 0.42
ALDH1A1 P00352 5/20 0.42
HPGD P15428 4/20 0.42
RAB9A P51151 3/20 0.42
GAA P10253 3/20 0.42
HSD17B10 Q99714 2/20 0.42
MAPT P10636 1/20 0.42
ALOX15 P16050 1/20 0.42
FNTA P49354 1/20 0.41
FNTB P49356 1/20 0.41
TSHR P16473 3/20 0.40
F2RL3 Q96RI0 1/20 0.39
TP53 P04637 2/20 0.38
KDM4E B2RXH2 3/20 0.38
NPC1 O15118 2/20 0.38
KMT2A Q03164 2/20 0.38
POLB P06746 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALOX5 P09917 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6167123 0.88 CYP19A1 (0.40) SMN1; SMN2ALDH1A1HPGDRAB9AGAA
Trifluoroacetic Acid SCHEMBL6167116 0.88 CYP19A1 (0.40) SMN1; SMN2ALDH1A1HPGDRAB9AGAA
Trifluoroacetic Acid SCHEMBL6164769 0.86 PRSS1 (0.45)
Trifluoroacetic Acid SCHEMBL6164778 0.86 PRSS1 (0.45)
Trifluoroacetic Acid SCHEMBL7101541 0.83 F10 (0.39)
Trifluoroacetic Acid SCHEMBL7101532 0.83 F10 (0.39)
Trifluoroacetic Acid SCHEMBL6165967 0.83 FNTA (0.39) SMN1; SMN2ALDH1A1HPGDRAB9AGAA
Trifluoroacetic Acid SCHEMBL6165974 0.83 FNTA (0.39) SMN1; SMN2ALDH1A1HPGDRAB9AGAA
Trifluoroacetic Acid SCHEMBL6163784 0.83 F10 (0.38)
Trifluoroacetic Acid SCHEMBL6163794 0.83 F10 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254136-A4 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD (KR) 2005-06-01 EP claimed
EP-1254136-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG Chem Investment, Ltd. (KR) 2002-11-06 EP claimed
WO-2001055146-A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF LG CHEM INVESTMENT LTD. (KR) 2001-08-02 WO claimed