SCHEMBL6173029

SCHEMBL6173029

COc1ccc2c(C(=O)c3ccc(CN4CCCC4)c(C)c3)c(-c3ccc(NC(C)=O)cc3)sc2c1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 14/20 0.57
ESR2 Q92731 14/20 0.57
ENPP3 O14638 3/20 0.51
ENPP1 P22413 3/20 0.51
MOK Q9UQ07 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7450865 0.93 ESR1 (0.56) ESR1ESR2ENPP3ENPP1
SCHEMBL6173615 0.89 ESR1 (0.68) ESR1ESR2
SCHEMBL6171805 0.88 ESR1 (0.60) ESR1ESR2ENPP3ENPP1
SCHEMBL6598683 0.86 ESR1 (0.70) ESR1ESR2ENPP3ENPP1
SCHEMBL6170231 0.85 ESR1 (0.56) ESR1ESR2ENPP3ENPP1
SCHEMBL7446013 0.82 ESR1 (0.71) ESR1ESR2ENPP3ENPP1
SCHEMBL7768048 0.82 F2 (0.58) ESR1ESR2
SCHEMBL6597618 0.80 ESR1 (0.49) ESR1ESR2ENPP3ENPP1
SCHEMBL7452932 0.80 ESR1 (0.76) ESR1ESR2ENPP3ENPP1
SCHEMBL7774305 0.78 ESR1 (0.79) ESR1ESR2ENPP3ENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027051-B1 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2005-01-05 EP disclosed
EP-0973517-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2002-07-24 EP disclosed
US-6391901-B1 Thrombin inhibitors ELI LILLY AND COMPANY 2002-05-21 US disclosed
US-6288105-B1 COMPOUNDS SUCH AS (S)-2-(4-((2-AMINO-3-HYDROXY-1-OXOPROPYL)AMINO)PHENYL)-6-HYDRO XY-3-(3-METHOXY-4-(1-PYRROLIDINYLMETHYL)BENZYL)BENZO(B)THIOPHE NE ELI LILLY AND COMPANY 2001-09-11 US disclosed
EP-0973517-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998048794-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed