SCHEMBL6176014

SCHEMBL6176014

C=C(Cl)C(=O)Nc1ccc2[nH]c(C(=O)Nc3cc(C(=O)Nc4cc(C(=O)Nc5cc(C(=O)NCCC(N)=O)n(C)c5)n(C)c4)n(C)c3)cc2c1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HRAS P01112 13/20 0.62
ESR1 P03372 13/20 0.62
ESR2 Q92731 13/20 0.62
TOP1 P11387 2/20 0.44
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
MAPT P10636 1/20 0.44
HIF1A Q16665 1/20 0.44
PYGL P06737 4/20 0.38
NHERF1 O14745 1/20 0.38
HDAC2 Q92769 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6966163 0.94 HRAS (0.71) HRASESR1ESR2TOP1KDM4E
Hydrochloric Acid SCHEMBL6974945 0.93 HRAS (0.71) HRASESR1ESR2TOP1KDM4E
SCHEMBL7128037 0.86 HRAS (0.57) HRASESR1ESR2TOP1KDM4E
SCHEMBL7116987 0.86 HRAS (0.57) HRASESR1ESR2TOP1KDM4E
SCHEMBL6969112 0.85 HRAS (0.69) HRASESR1ESR2TOP1KDM4E
Hydrochloric Acid SCHEMBL6978383 0.85 HRAS (0.69) HRASESR1ESR2TOP1KDM4E
SCHEMBL6176871 0.83 HRAS (0.59) HRASESR1ESR2TOP1KDM4E
SCHEMBL6176114 0.79 HRAS (0.52) HRASESR1ESR2TOP1KDM4E
SCHEMBL6976518 0.79 HRAS (0.54) HRASESR1ESR2TOP1KDM4E
Hydrochloric Acid SCHEMBL6968970 0.79 HRAS (0.54) HRASESR1ESR2TOP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1064281-B1 BENZOHETEROCYCLIC DISTAMYCIN DERIVATIVES, PROCESS FOR PREPARING THEM, AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-05-25 EP claimed
US-6458768-B1 ANTITUMOR AGENTS THAT CAN BE FORMULATED WITH A COMPOUND ALTERNATIVELY, CAN BE ADMINISTERED IN A MIXTURE OF DRUGS PHARMACIA & UPJOHN, S.P.A. (IT) 2002-10-01 US claimed
EP-1064281-B1 BENZOHETEROCYCLIC DISTAMYCIN DERIVATIVES, PROCESS FOR PREPARING THEM, AND THEIR USE AS ANTITUMOR AGENTS PHARMACIA ITALIA SPA (IT) 2005-05-25 EP disclosed
US-6458768-B1 ANTITUMOR AGENTS THAT CAN BE FORMULATED WITH A COMPOUND ALTERNATIVELY, CAN BE ADMINISTERED IN A MIXTURE OF DRUGS PHARMACIA & UPJOHN, S.P.A. (IT) 2002-10-01 US disclosed