SCHEMBL6182149

SCHEMBL6182149

[CH2]COCCOc1ncccc1OCCOc1nccnc1N1CCNC[C@H]1C

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 13/20 0.40
HTR2A P28223 9/20 0.40
HTR2B P41595 8/20 0.40
KCNH2 Q12809 1/20 0.38
LATS1 O95835 1/20 0.33
HTR1A P08908 1/20 0.33
SLC6A2 P23975 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
GSK3B P49841 2/20 0.32
SSTR1 P30872 1/20 0.32
SSTR4 P31391 1/20 0.32
CHRNB4 P30926 1/20 0.31
CHRNA3 P32297 1/20 0.31
ROCK1 Q13464 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL906101 0.90 HTR2C (0.40) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL237951 0.89 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL2639684 0.89 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL905805 0.89 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2LATS1
SCHEMBL4313537 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL2639295 0.88 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL906015 0.86 HTR2C (0.40) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL6047120 0.86 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL237834 0.86 HTR2C (0.42) HTR2CHTR2AHTR2BKCNH2HTR1A
SCHEMBL905949 0.86 HTR2C (0.43) HTR2CHTR2AHTR2BKCNH2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1513831-A1 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Biovitrum AB (SE) 2005-03-16 EP claimed
WO-2004000830-A1 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2003-12-31 WO claimed
EP-1513831-A1 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Biovitrum AB (SE) 2005-03-16 EP disclosed
WO-2004000830-A1 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2003-12-31 WO disclosed