SCHEMBL6183161

SCHEMBL6183161

CCOC(=O)N1c2cc(C(F)(F)F)c(OC)cc2C(N(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)C(=O)OC)CC1C1CC1

nearest known ligand 0.60

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CETP P11597 20/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6183155 1.00 CETP (0.60) CETP
SCHEMBL6590043 0.90 CETP (0.63) CETP
SCHEMBL6590045 0.90 CETP (0.63) CETP
SCHEMBL6179751 0.90 CETP (0.65) CETP
SCHEMBL6179756 0.90 CETP (0.65) CETP
SCHEMBL6183580 0.89 CETP (0.64) CETP
SCHEMBL6183577 0.89 CETP (0.64) CETP
SCHEMBL6184660 0.88 CETP (0.56) CETP
SCHEMBL6184663 0.88 CETP (0.56) CETP
SCHEMBL6182477 0.88 CETP (0.61) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1607389-A1 4-protected-amino-2-substituted-1,2,3,4-tetrahydroquinolines as intermediates for CETP inhibitors Pfizer Products Inc. (US) 2005-12-21 EP disclosed
EP-1114031-B1 4-CARBOXYAMINO-2-SUBSTITUTED-1,2,3,4-TETRAHYDROQUINOLINES AS CETP INHIBITORS PFIZER PROD INC (US) 2005-06-15 EP disclosed
US-6586448-B1 Cholesteryl ester transfer protein inhibitors used as antilipemic agents for prophylaxis of cardiovascular disorders PFIZER INC. 2003-07-01 US disclosed
US-6197786-B1 ANTICHOLESTEROL AGENTS PFIZER INC 2001-03-06 US disclosed