SCHEMBL6183865

SCHEMBL6183865

COC(=O)N(Cc1cc(C(F)(F)F)cc(C(F)(F)F)c1)[C@H]1C[C@@H](C2CC2)N(C(=O)OC(C)C)c2cc3c(cc21)CCC3

nearest known ligand 0.57

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
CETP P11597 20/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6183870 1.00 CETP (0.57) CETP
SCHEMBL6182060 0.95 CETP (0.51) CETP
SCHEMBL6182054 0.95 CETP (0.51) CETP
SCHEMBL6185569 0.93 CETP (0.51) CETP
SCHEMBL6185572 0.93 CETP (0.51) CETP
SCHEMBL6182479 0.91 CETP (0.61) CETP
SCHEMBL6182477 0.91 CETP (0.61) CETP
SCHEMBL6181519 0.91 CETP (0.54) CETP
SCHEMBL6182097 0.91 CETP (0.52) CETP
SCHEMBL6181522 0.91 CETP (0.54) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1607389-A1 4-protected-amino-2-substituted-1,2,3,4-tetrahydroquinolines as intermediates for CETP inhibitors Pfizer Products Inc. (US) 2005-12-21 EP disclosed
EP-1114031-B1 4-CARBOXYAMINO-2-SUBSTITUTED-1,2,3,4-TETRAHYDROQUINOLINES AS CETP INHIBITORS PFIZER PROD INC (US) 2005-06-15 EP disclosed
US-6586448-B1 Cholesteryl ester transfer protein inhibitors used as antilipemic agents for prophylaxis of cardiovascular disorders PFIZER INC. 2003-07-01 US disclosed
US-6197786-B1 ANTICHOLESTEROL AGENTS PFIZER INC 2001-03-06 US disclosed