SCHEMBL6184872

SCHEMBL6184872

O=C1NC(=O)C(=Cc2ccc(-c3cccc(N(C(=O)O)c4ccccc4)c3)cc2)S1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 5/20 0.55
PIM2 Q9P1W9 5/20 0.55
PIM3 Q86V86 1/20 0.55
NAT1 P18440 1/20 0.53
GSK3B P49841 1/20 0.53
MEN1 O00255 1/20 0.53
POLB P06746 1/20 0.53
KMT2A Q03164 1/20 0.53
HPGD P15428 4/20 0.51
AKR1B1 P15121 4/20 0.50
GLS O94925 1/20 0.50
GLS2 Q9UI32 1/20 0.50
PTPN1 P18031 2/20 0.49
CISD1 Q9NZ45 2/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5386767 0.86 GSK3B (0.59) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL1248782 0.81 PIM1 (0.83) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL1248780 0.81 PIM1 (0.83) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL12891790 0.81 PIM1 (0.83) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL6185404 0.80 HPGD (0.53) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL6204139 0.80 GSK3B (0.52) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL6185401 0.80 HPGD (0.53) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL6204137 0.80 GSK3B (0.52) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL6202184 0.80 PIM1 (0.76) PIM1PIM2PIM3NAT1GSK3B
SCHEMBL6184899 0.79 PIK3CG (0.67) PIM1PIM2PIM3NAT1GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6927228-B2 Biphenyl compounds usefuf in treatment of human and veterinary medicines such as dermatology, cardivovascular diseases, immune diseases or diseases associated with lipid metabolisms, or in cosmetic formulation GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-09 US claimed
EP-1309575-B1 BIPHENYL DERIVATIVES AND THEIR USE AS PPAR-GAMMA RECEPTOR ACTIVATORS GALDERMA RES & DEV (FR) 2005-06-08 EP claimed
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2004-02-26 US claimed
US-6927228-B2 Biphenyl compounds usefuf in treatment of human and veterinary medicines such as dermatology, cardivovascular diseases, immune diseases or diseases associated with lipid metabolisms, or in cosmetic formulation GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-09 US disclosed
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors PPARG, PPARA, PPARD PIM1 4083/4885PIM2 4126/4885PIM3 4524/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.