SCHEMBL6185166

SCHEMBL6185166

CN(Cc1cccc(-c2ccc(C=C3SC(=O)NC3=O)cc2)c1)C(=O)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 5/20 0.51
HSD17B1 P14061 4/20 0.51
PTPN1 P18031 3/20 0.51
HPGD P15428 6/20 0.50
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
PIM1 P11309 1/20 0.47
PIM3 Q86V86 1/20 0.47
PIM2 Q9P1W9 1/20 0.47
POLB P06746 1/20 0.47
GSK3B P49841 1/20 0.47
NAT1 P18440 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6185163 1.00 HSD17B2 (0.51) HSD17B2HSD17B1PTPN1HPGDMEN1
SCHEMBL6184406 0.94 MEN1 (0.53) HSD17B2HSD17B1PTPN1HPGDMEN1
SCHEMBL6184404 0.94 MEN1 (0.53) HSD17B2HSD17B1PTPN1HPGDMEN1
SCHEMBL5397253 0.90 MEN1 (0.53) PTPN1HPGDMEN1KMT2APIM1
SCHEMBL5397249 0.90 MEN1 (0.53) PTPN1HPGDMEN1KMT2APIM1
SCHEMBL6183613 0.89 PTPN1 (0.50) PTPN1HPGDMEN1KMT2APIM1
SCHEMBL6183616 0.89 PTPN1 (0.50) PTPN1HPGDMEN1KMT2APIM1
SCHEMBL6183241 0.87 PTPN1 (0.48) PTPN1HPGDMEN1KMT2APIM1
SCHEMBL6183238 0.87 PTPN1 (0.48) PTPN1HPGDMEN1KMT2APIM1
SCHEMBL1750572 0.87 PTPN1 (0.48) PTPN1HPGDPIM1PIM3PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6927228-B2 Biphenyl compounds usefuf in treatment of human and veterinary medicines such as dermatology, cardivovascular diseases, immune diseases or diseases associated with lipid metabolisms, or in cosmetic formulation GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2005-08-09 US disclosed
EP-1309575-B1 BIPHENYL DERIVATIVES AND THEIR USE AS PPAR-GAMMA RECEPTOR ACTIVATORS GALDERMA RES & DEV (FR) 2005-06-08 EP disclosed
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors GALDERMA RESEARCH & DEVELOPMENT S.N.C. (FR) 2004-02-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040039038-A1 Biaromatic compound activators of PPARy-type receptors PPARG, PPARA, PPARD HSD17B2 368/4885HSD17B1 275/4885PTPN1 1579/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.