SCHEMBL6189655

SCHEMBL6189655

CCN(CCCOc1ccc(N=C=S)cc1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.43
NPC1 O15118 2/20 0.43
LMNA P02545 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43
BCHE P06276 3/20 0.40
ACHE P22303 3/20 0.40
PPARA Q07869 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HCRTR1 O43613 1/20 0.39
HCRTR2 O43614 1/20 0.39
PRSS1 P07477 1/20 0.39
ACR P10323 1/20 0.39
PPARG P37231 1/20 0.39
ALDH1A1 P00352 1/20 0.39
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180008 0.84 PPARA (0.39) HSD17B10NPC1LMNAALOX15TSHR
SCHEMBL2481800 0.83 NPC1 (0.44) HSD17B10NPC1LMNAALOX15TSHR
SCHEMBL6181833 0.78 MEN1 (0.36) HSD17B10PPARAMEN1KMT2APPARG
SCHEMBL3597778 0.77 KDM4E (0.59) ALDH1A1
SCHEMBL9362384 0.76 CYP2C9 (0.51) HSD17B10NPC1LMNAALOX15TSHR
SCHEMBL3609469 0.76 EBP (0.54) MEN1KMT2A
SCHEMBL2480421 0.74 BCHE (0.41) HSD17B10NPC1LMNAALOX15TSHR
SCHEMBL6192856 0.72 P2RY6 (0.48) HSD17B10NPC1ALOX15TSHRMAPK1
SCHEMBL631842 0.72 HRH3 (0.54) ALDH1A1
SCHEMBL24184660 0.71 CYP1A2 (0.46) LMNATSHRALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1507530-B1 DIAMINOTHIAZOLES AND USE THEREOF AS CDK4 INHIBITORS HOFFMANN LA ROCHE (CH) 2005-11-02 EP disclosed