SCHEMBL6199477

SCHEMBL6199477

CCCCCCCCCc1ccc(CN2CCC(O)(P(=O)(O)O)C2)cc1

nearest known ligand 0.62

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 13/20 0.62
S1PR3 Q99500 9/20 0.62
S1PR4 O95977 6/20 0.62
S1PR5 Q9H228 5/20 0.62
ENPP2 Q13822 1/20 0.48
HRH3 Q9Y5N1 3/20 0.47
THRA P10827 1/20 0.43
THRB P10828 1/20 0.43
S1PR2 O95136 3/20 0.42
SPHK1 Q9NYA1 2/20 0.42
SPHK2 Q9NRA0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13937984 0.85 S1PR5 (0.56) S1PR1S1PR3S1PR4S1PR5
SCHEMBL13937989 0.85 S1PR5 (0.56) S1PR1S1PR3S1PR4S1PR5THRA
SCHEMBL13937991 0.82 S1PR1 (0.53) S1PR1S1PR3S1PR4S1PR5S1PR2
SCHEMBL6181254 0.80 S1PR1 (0.57) S1PR1S1PR3S1PR4S1PR5HRH3
SCHEMBL6179863 0.80 S1PR1 (0.57) S1PR1S1PR3S1PR4S1PR5HRH3
SCHEMBL13937987 0.79 S1PR1 (0.51) S1PR1S1PR3S1PR4S1PR5S1PR2
SCHEMBL6179864 0.77 S1PR1 (0.48) S1PR1S1PR3S1PR4S1PR5HRH3
SCHEMBL6362290 0.77 S1PR1 (0.48) S1PR1S1PR3S1PR4S1PR5HRH3
SCHEMBL3909200 0.76 S1PR1 (0.50) S1PR1S1PR3S1PR4S1PR5HRH3
SCHEMBL3909199 0.76 S1PR1 (0.50) S1PR1S1PR3S1PR4S1PR5HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7479504-B2 Edg receptor agonists MERCK & CO., INC. (US) 2009-01-20 US disclosed
US-7479504-B2 Edg receptor agonists MERCK & CO., INC. (US) 2009-01-20 US disclosed
EP-1470137-A4 EDG RECEPTOR AGONISTS MERCK & CO INC (US) 2005-06-15 EP disclosed
EP-1470137-A1 EDG RECEPTOR AGONISTS Merck & Co., Inc. (US) 2004-10-27 EP disclosed
WO-2003062252-A1 EDG RECEPTOR AGONISTS MERCK & CO., INC. (US) 2003-07-31 WO disclosed