SCHEMBL6202054

SCHEMBL6202054

c1cnc2ccc(OCCn3ccc4ccc5c(c43)CCNCC5)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 7/20 0.40
CYP2D6 P10635 1/20 0.39
HRH1 P35367 1/20 0.38
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
MCL1 Q07820 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGAV P06756 1/20 0.35
CHKA P35790 1/20 0.34
HTR2A P28223 2/20 0.33
HTR2C P28335 2/20 0.33
HTR2B P41595 2/20 0.33
DRD3 P35462 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6097921 0.81 HRH3 (0.40) HRH3HRH1MCL1HTR2AHTR2C
SCHEMBL6097603 0.80 MAPT (0.41) HRH3HTR2AHTR2CHTR2BKDM4E
SCHEMBL6099299 0.77 MCL1 (0.43) HRH3HRH1MCL1HTR2AHTR2C
SCHEMBL6099897 0.76 KDM4E (0.41) HRH3CYP2D6HTR2AHTR2CHTR2B
SCHEMBL6098861 0.76 HIF1A (0.43) SLC6A2HTR2AHTR2CHTR2BKDM4E
SCHEMBL6096642 0.72 HRH3 (0.46) HRH3MCL1
SCHEMBL6482908 0.67 DRD3 (0.42) HRH3HRH1SLC6A2SLC6A4DRD3
SCHEMBL6474621 0.66 DRD3 (0.42) HTR2ADRD3
SCHEMBL6358473 0.66 MCL1 (0.43) CYP2D6SLC6A2SLC6A4MCL1KDM4E
SCHEMBL6474563 0.66 DRD3 (0.45) DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406902-B1 HEXAHYDROAZEPINO[4,5-G]INDOLES AND INDOLINES AS 5-HT RECEPTOR LIGANDS PHARMACIA & UPJOHN CO LLC (US) 2005-10-19 EP claimed