SCHEMBL6203400

SCHEMBL6203400

CCCCNCc1c(-c2ccccc2)nc2ccccc2c1OC(=O)N[C@@H](C)C1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 13/20 0.53
TACR2 P21452 12/20 0.53
OPRM1 P35372 6/20 0.51
CYP2C9 P11712 2/20 0.44
NTRK1 P04629 1/20 0.43
EPHX2 P34913 2/20 0.41
TRPV4 Q9HBA0 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201095 0.83 TACR3 (0.54) TACR3TACR2OPRM1CYP2C9NTRK1
SCHEMBL6202146 0.80 TACR2 (0.59) TACR3TACR2OPRM1TRPV4
SCHEMBL6201403 0.79 TACR2 (0.62) TACR3TACR2OPRM1TRPV4
SCHEMBL6245604 0.78 TACR2 (0.62) TACR3TACR2OPRM1TRPV4
SCHEMBL6202395 0.78 TACR2 (0.62) TACR3TACR2OPRM1TRPV4
SCHEMBL6199955 0.78 TACR2 (0.66) TACR3TACR2OPRM1TRPV4
SCHEMBL6200693 0.78 TACR2 (0.59) TACR3TACR2OPRM1CYP2C9NTRK1
SCHEMBL6203216 0.78 TACR2 (0.63) TACR3TACR2OPRM1TRPV4
SCHEMBL6202169 0.77 TACR2 (0.74) TACR3TACR2OPRM1TRPV4
SCHEMBL6197279 0.77 TACR2 (0.54) TACR3TACR2OPRM1CYP2C9NTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377567-B1 QUINOLINE-4-CARBOXAMIDE DERIVATIVES AS NK-3 AND NK-2 RECEPTOR ANTAGONISTS GLAXOSMITHKLINE SPA (IT) 2005-12-21 EP claimed