SCHEMBL6203575

SCHEMBL6203575

COc1ccc(F)c2c1CC(CN1CC(C)(C)Cn3c1nc(-c1ccncn1)cc3=O)CO2

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.40
CYP2D6 P10635 7/20 0.40
CYP1A2 P05177 5/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6201903 0.83 GSK3B (0.40) GSK3BCYP2D6CYP1A2
SCHEMBL6630868 0.79 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL6628760 0.79 GSK3B (0.41) GSK3BCYP2D6CYP1A2
SCHEMBL5102710 0.77 GSK3B (0.44) GSK3BCYP2D6CYP1A2
SCHEMBL3563586 0.76 GSK3B (0.46) GSK3BCYP2D6CYP1A2
SCHEMBL5151545 0.75 GSK3B (0.39) GSK3BCYP2D6CYP1A2
SCHEMBL6204428 0.74 GSK3B (0.40) GSK3BCYP2D6CYP1A2
SCHEMBL3573554 0.74 GSK3B (0.50) GSK3BCYP2D6CYP1A2
SCHEMBL3566745 0.73 GSK3B (0.46) GSK3BCYP2D6CYP1A2
SCHEMBL5095642 0.73 GSK3B (0.43) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1480983-B1 HETEROARYL SUBSTITUTED 2-PYRIDINYL AND 2-PYRIMIDINYL-6,7,8,9-TETRAHYDROPYDIMIDO[1,2-A]PYRIMIDIN-4-ONE DERIVATIVES SANOFI AVENTIS (FR) 2005-11-09 EP disclosed
EP-1480983-A1 HETEROARYL SUBSTITUTED 2-PYRIDINYL AND 2-PYRIMIDINYL-6,7,8,9-TETRAHYDROPYDIMIDO[1,2-A]PYRIMIDIN-4-ONE DERIVATIVES Sanofi-Aventis (FR) 2004-12-01 EP disclosed
WO-2003072579-A1 HETEROARYL SUBSTITUTED 2-PYRIDINYL AND 2-PYRIMIDINYL -6,7,8,9- TETRAHYDROPYRIMIDO[1,2-a] PYRIMIDIN-4-ONE DERIVATIVES SANOFI-AVENTIS (FR) 2003-09-04 WO disclosed