SCHEMBL6203679

SCHEMBL6203679

O=C1NCCn2c(-c3ccncc3)nc3cccc1c32

nearest known ligand 0.83

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 20/20 0.83
PARP2 Q9UGN5 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6199272 0.97 PARP1 (0.80) PARP1PARP2
SCHEMBL831830 0.91 PARP1 (1.00) PARP1
SCHEMBL12750571 0.89 PARP1 (1.00) PARP1PARP2
SCHEMBL12750579 0.88 PARP1 (0.80) PARP1PARP2
SCHEMBL7158077 0.88 PARP1 (1.00) PARP1
SCHEMBL20570669 0.88 PARP1 (0.80) PARP1PARP2
SCHEMBL6200038 0.88 PARP1 (0.80) PARP1
SCHEMBL7162347 0.86 PARP1 (0.78) PARP1PARP2
SCHEMBL7164754 0.86 PARP1 (0.77) PARP1PARP2
SCHEMBL6203088 0.85 PARP1 (0.77) PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208104-B1 TRICYCLIC INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASES AGOURON PHARMA (US) 2005-01-19 EP disclosed
US-6548494-B1 3,4-dihydro-2H-(1,4)diazepino(6,7,1-hi)indol-1-one or 1-thione derivatives where indole C3 could also be N; use treating cancers as well as stroke, head trauma, and neurodegenerative diseases AGOURON PHARMACEUTICALS, INC. 2003-04-15 US disclosed
EP-1222191-A2 BENZODIAZEPIN DERIVATIVES, THE PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-07-17 EP disclosed
WO-2001023386-A2 BENZODIAZEPIN DERIVATIVES, THE PRODUCTION AND USE THEREOF BASF AKTIENGESELLSCHAFT (DE) 2001-04-05 WO disclosed