SCHEMBL6205522

SCHEMBL6205522

CCCCOCCOc1ccc(-c2cc3c4c(c2)OCCN4CCC/C(C(=O)OCC)=C\3)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.41
CCR5 P51681 11/20 0.41
CCR2 P41597 2/20 0.39
CCR7 P32248 1/20 0.39
KCNH2 Q12809 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
RARA P10276 1/20 0.38
CCR3 P51677 1/20 0.37
CCR4 P51679 1/20 0.37
POLB P06746 1/20 0.37
HRH2 P25021 1/20 0.35
HRH1 P35367 1/20 0.35
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205525 1.00 RARB (0.41) RARBCCR5CCR2CCR7KCNH2
SCHEMBL6204657 0.91 RARB (0.48) RARBCCR5CCR2CCR7RARA
SCHEMBL6204659 0.91 RARB (0.48) RARBCCR5CCR2CCR7RARA
SCHEMBL5940268 0.88 RARB (0.44) RARBCCR5CCR2CCR7KCNH2
SCHEMBL5940270 0.88 RARB (0.44) RARBCCR5CCR2CCR7KCNH2
SCHEMBL5940260 0.87 RARB (0.44) RARBCCR5CCR2CCR7KCNH2
SCHEMBL5940257 0.87 RARB (0.44) RARBCCR5CCR2CCR7KCNH2
SCHEMBL5940261 0.85 RARB (0.44) RARBCCR5CCR2CCR7KCNH2
SCHEMBL3459772 0.83 RARB (0.45) RARBCCR5CCR2CCR7KCNH2
SCHEMBL3459770 0.83 RARB (0.45) RARBCCR5CCR2CCR7KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1593681-A1 TRICYCLIC COMPOUND, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Pharmaceutical Company Limited (JP) 2005-11-09 EP disclosed