SCHEMBL6207836

SCHEMBL6207836

COCCCNc1nnc(-c2ccc(F)c(F)c2Nc2ccc(I)cc2F)o1.Fc1cc(I)ccc1Nc1c(-c2nnc(NCCN3CCOCC3)o2)ccc(F)c1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 15/20 0.46
KCNH2 Q12809 14/20 0.46
CHRNA1 P02708 2/20 0.44
CYP3A4 P08684 2/20 0.44
CHRNB2 P17787 2/20 0.44
CHRNA4 P43681 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
MAP2K1 Q02750 2/20 0.43
MAP2K2 P36507 1/20 0.43
MAP3K8 P41279 1/20 0.39
CYP2D6 P10635 1/20 0.39
CSF1R P07333 1/20 0.39
PIK3CD O00329 1/20 0.37
PIK3R1 P27986 1/20 0.37
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
PIM1 P11309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207045 0.92 MAP2K2 (0.47) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
SCHEMBL29371646 0.92 MAP2K2 (0.47) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
Hydrochloric Acid SCHEMBL6206110 0.90 CHRNA7 (0.48) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
SCHEMBL6406299 0.90 PIM1 (0.44) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
SCHEMBL6205441 0.85 CHRNA7 (0.46) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
SCHEMBL6208038 0.85 PIM1 (0.45) MAP2K1MAP2K2PIM1CAMK2B
SCHEMBL15598681 0.84 CHRNA7 (0.44) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
SCHEMBL6399647 0.83 CHRNA7 (0.48) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
SCHEMBL6399220 0.83 CHRNA7 (0.43) CHRNA7KCNH2CHRNA1CYP3A4CHRNB2
SCHEMBL6399299 0.82 PIM1 (0.41) MAP2K1MAP2K2PIM1CAMK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1578736-A1 MEK INHIBITING OXA- AND THIA-DIAZOL-2-YL-PHENYLAMINE DERIVATIVES Warner-Lambert Company LLC (US) 2005-09-28 EP claimed
WO-2004056789-A1 MEK INHIBITING OXA- AND THIA-DIAZOL-2-YL PHENYLAMINE DERIVATES WARNER-LAMBERT COMPANY LLC (US) 2004-07-08 WO claimed