SCHEMBL6207912

SCHEMBL6207912

COc1cccc(-c2ncoc2-c2ccc(O)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.50
ABL1 P00519 3/20 0.49
ABCB1 P08183 3/20 0.49
BCR P11274 3/20 0.49
VCP P55072 1/20 0.47
NOTUM Q6P988 1/20 0.46
DYRK1A Q13627 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
GSK3B P49841 1/20 0.44
PPARG P37231 1/20 0.43
PPARD Q03181 1/20 0.43
PPARA Q07869 1/20 0.43
HSD17B10 Q99714 2/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
CYP3A4 P08684 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6539721 0.84 ESR2 (0.55) ABL1ABCB1BCRGSK3BKDM4E
2-Mercaptoethanol SCHEMBL11751369 0.82 HSD17B10 (0.47) NOTUMDYRK1ACLK4GSK3BHSD17B10
SCHEMBL11751584 0.80 KDM4E (0.47) NOTUMGSK3BHSD17B10KDM4EMEN1
SCHEMBL27934283 0.77 CYP1A1 (0.45) ABL1ABCB1BCRGSK3BKDM4E
SCHEMBL27840064 0.76 MAPK14 (0.51) CLK4GSK3BKDM4EMEN1KMT2A
SCHEMBL24177866 0.76 ABL1 (0.79) FYNABL1ABCB1BCRMEN1
SCHEMBL1513611 0.76 ABL1 (0.79) FYNABL1ABCB1BCRMEN1
SCHEMBL11752862 0.75 KDM4E (0.50) NOTUMGSK3BHSD17B10KDM4EMEN1
SCHEMBL27820747 0.74 CYP1A1 (0.45) ABL1ABCB1BCRDYRK1ACLK4
SCHEMBL15665148 0.73 CYP1A1 (0.42) HSD17B10KDM4ECYP3A4ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583749-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE Astellas Pharma Inc. (JP) 2005-10-12 EP disclosed
WO-2004065374-A1 OXAZOLE DERIVATIVES AS INHIBITORS OF CYCLOOXYGENASE ASTELLAS PHARMA INC. (JP) 2004-08-05 WO disclosed