SCHEMBL6208907

SCHEMBL6208907

CC1=C(c2ccc(C(=O)N3Cc4ccc(OC(=O)N(C)Cc5cccnc5)n4Cc4ccccc43)cc2C)CCC[C@H]1O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 3/20 0.37
AVPR2 P30518 8/20 0.36
POLB P06746 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PDK1 Q15118 3/20 0.34
PDK2 Q15119 3/20 0.34
PDK3 Q15120 3/20 0.34
PDK4 Q16654 3/20 0.34
STAT3 P40763 1/20 0.34
BRD4 O60885 1/20 0.33
OXTR P30559 1/20 0.33
ROCK2 O75116 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6207415 0.78 AVPR2 (0.39) AVPR1AAVPR2POLBHSD17B10STAT3
SCHEMBL6207413 0.77 AVPR1A (0.38) AVPR1AAVPR2POLBHSD17B10OXTR
SCHEMBL5117311 0.77 AVPR2 (0.43) AVPR1AAVPR2
SCHEMBL5117936 0.77 AVPR2 (0.43) AVPR1AAVPR2
SCHEMBL5891244 0.74 AVPR2 (0.46) AVPR1AAVPR2PDK1PDK2PDK3
SCHEMBL5111220 0.74 AVPR2 (0.46) AVPR1AAVPR2BRD4OXTR
SCHEMBL5143793 0.74 AVPR2 (0.46) AVPR1AAVPR2BRD4OXTR
SCHEMBL5119243 0.74 AVPR2 (0.46) AVPR1AAVPR2BRD4OXTR
SCHEMBL6068860 0.73 AVPR1A (0.57) AVPR1AAVPR2OXTR
SCHEMBL5106769 0.73 AVPR1A (0.57) AVPR1AAVPR2OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381607-B1 NOVEL PYRIDINE- AND CYCLOHEXENYL-COMPRISING PYRROLOBENZODIAZEPINE-CARBOXAMIDES AND DERIVATIVES THEREOF; TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS WYETH CORP (US) 2005-10-26 EP claimed