SCHEMBL6217992

SCHEMBL6217992

COc1ccc(C(=O)c2nc(C(F)(F)F)nc3ccsc23)s1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 20/20 0.64
ADORA1 P30542 14/20 0.64
ADORA2B P29275 5/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6861124 0.85 ADORA2A (0.71) ADORA2AADORA1ADORA2B
SCHEMBL6859592 0.83 ADORA2A (0.70) ADORA2AADORA1ADORA2B
SCHEMBL6216685 0.82 ADORA2A (0.72) ADORA2AADORA1ADORA2B
SCHEMBL6217941 0.82 ADORA2A (0.64) ADORA2AADORA1ADORA2B
SCHEMBL6852945 0.80 ADORA2A (0.71) ADORA2AADORA1ADORA2B
SCHEMBL6217242 0.78 ADORA2A (1.00) ADORA2AADORA1
SCHEMBL6852837 0.76 ADORA2A (0.76) ADORA2AADORA1ADORA2B
SCHEMBL6214990 0.75 ADORA2A (1.00) ADORA2AADORA1ADORA2B
SCHEMBL6852789 0.75 ADORA2A (0.68) ADORA2AADORA1ADORA2B
SCHEMBL6859881 0.75 ADORA2A (0.70) ADORA2AADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1192164-B1 THIENO- AND FUROPYRIMIDINE DERIVATIVES AS A2A-RECEPTOR ANTAGONISTS VERNALIS RES LTD (GB) 2005-08-17 EP disclosed
US-6787541-B1 MOVEMENT DISORDERS, PARKINSON'S DISEASE VERNALIS RESEARCH LIMITED (GB) 2004-09-07 US disclosed