SCHEMBL6224980

SCHEMBL6224980

O=C(Nc1cc(F)cc(F)c1O)NC12CC3CC(CC(C3)C1)C2.O=C(Nc1ccc(Oc2ccccc2)cc1)Nc1cc(F)cc(F)c1O.O=C(Nc1ccccc1)Nc1cc(F)cc(F)c1O

nearest known ligand 0.69

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 19/20 0.69
RAF1 P04049 1/20 0.49
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA9 Q16790 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6249917 0.91 EPHX2 (0.66) EPHX2RAF1CA12CA1CA2
SCHEMBL6228091 0.89 EPHX2 (0.71) EPHX2
SCHEMBL4345603 0.85 CA12 (0.54) CA12CA1CA2CA9
SCHEMBL6255295 0.84 EPHX2 (0.62) EPHX2
SCHEMBL6224093 0.83 EPHX2 (0.69) EPHX2RAF1
SCHEMBL4347622 0.83 EPHX2 (0.60) EPHX2
SCHEMBL6250598 0.82 EPHX2 (0.76) EPHX2RAF1CA12CA1CA2
SCHEMBL6225545 0.82 EPHX2 (0.76) EPHX2RAF1CA12CA1CA2
SCHEMBL6226060 0.81 EPHX2 (0.65) EPHX2RAF1
SCHEMBL6680961 0.80 EPHX2 (0.61) EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539683-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS Jerini AG (DE) 2005-06-15 EP claimed
WO-2004026815-A2 PHENOL DERIVATIVES AND THEIR USE AS ROTAMASE INHIBITORS JERINI AG (DE) 2004-04-01 WO claimed