SCHEMBL6232111

SCHEMBL6232111

CC(C)CCn1c(=O)c(C2=NS(=O)(=O)c3cc([O])ccc3N2)c(O)c2ccccc21

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.67
HSD17B10 Q99714 1/20 0.67
CYP2C9 P11712 3/20 0.50
NR1I2 O75469 1/20 0.50
KDM4E B2RXH2 7/20 0.39
ALDH1A1 P00352 6/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 3/20 0.39
NPC1 O15118 1/20 0.38
PLK1 P53350 1/20 0.38
APOBEC3G Q9HC16 1/20 0.38
XBP1 P17861 1/20 0.38
NPSR1 Q6W5P4 2/20 0.37
RXFP1 Q9HBX9 1/20 0.37
MAPT P10636 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6236195 0.92 MAPK1 (0.68) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6235524 0.91 MAPK1 (0.67) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6236122 0.91 MAPK1 (0.67) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6235167 0.90 MAPK1 (0.66) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6741396 0.90 MAPK1 (0.66) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6232243 0.90 MAPK1 (0.66) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6236792 0.90 MAPK1 (0.66) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL12403127 0.90 MAPK1 (0.82) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6232841 0.90 HSD17B10 (0.65) MAPK1HSD17B10CYP2C9NR1I2KDM4E
SCHEMBL6232817 0.89 MAPK1 (0.64) MAPK1HSD17B10CYP2C9NR1I2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401443-A4 NOVEL ANTI-INFECTIVES SMITHKLINE BEECHAM CORP (US) 2005-10-26 EP disclosed
EP-1401443-A1 NOVEL ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2004-03-31 EP disclosed
WO-2002098424-A1 NOVEL ANTI-INFECTIVES SMITHKLINE BEECHAM CORPORATION (US) 2002-12-12 WO disclosed