SCHEMBL6232756

SCHEMBL6232756

CC(C)[C@H](O)C(=O)NCCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.59
CYP2D6 P10635 1/20 0.59
CYP2C9 P11712 1/20 0.59
CYP2C19 P33261 1/20 0.59
POLB P06746 1/20 0.59
MEN1 O00255 1/20 0.56
TSHR P16473 1/20 0.56
LAP3 P28838 2/20 0.54
ANPEP P15144 2/20 0.54
RNPEP Q9H4A4 1/20 0.54
DNPEP Q9ULA0 1/20 0.54
CA12 O43570 1/20 0.53
CA2 P00918 1/20 0.53
CA9 Q16790 1/20 0.53
EPHX1 P07099 1/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
ALDH1A1 P00352 1/20 0.51
HPGD P15428 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10635162 0.90 POLB (0.61) KMT2ACYP2D6CYP2C9CYP2C19POLB
SCHEMBL9192833 0.90 POLB (0.61) KMT2ACYP2D6CYP2C9CYP2C19POLB
SCHEMBL31126659 0.86 KMT2A (0.63) KMT2ACYP2D6CYP2C9CYP2C19POLB
SCHEMBL2275011 0.85 KMT2A (0.61) KMT2ACYP2D6CYP2C9CYP2C19POLB
SCHEMBL20589831 0.84 KMT2A (0.55) KMT2ACYP2D6CYP2C9CYP2C19POLB
SCHEMBL7866857 0.84 KMT2A (0.81) KMT2ACYP2D6CYP2C9CYP2C19POLB
Hydrochloric Acid SCHEMBL27729415 0.83 KMT2A (0.78) KMT2ACYP2D6CYP2C9CYP2C19POLB
SCHEMBL25681471 0.83 KMT2A (0.61) KMT2AMEN1TSHRCA12CA2
SCHEMBL10492080 0.82 POLB (0.61) KMT2ACYP2D6CYP2C9CYP2C19POLB
SCHEMBL9188615 0.82 POLB (0.54) KMT2ACYP2D6CYP2C9CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1049481-B1 SYNTHETIC ANTINEOPLASTIC AGENTS DERIVED FROM DOLASTATIN 15 AND METHODS OF MAKING SAME UNIV ARIZONA (US) 2005-04-20 EP disclosed
US-6686445-B1 ESTERIFICATION OF 2-HYDROXYISOVALERIC ACID AND TBOC-L-PROLINE; SALT FORMATION WITH TRIFLUORACETIC ACID; DEPROTECTING AND REACTING WITH N,N'-DIMETHYLVALINE ARIZONA BOARD OF REGENTS, ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY 2004-02-03 US disclosed
EP-1049481-A4 SYNTHETIC ANTINEOPLASTIC AGENTS DERIVED FROM DOLASTATIN 15 AND METHODS OF MAKING SAME UNIV ARIZONA (US) 2001-09-12 EP disclosed
EP-1049481-A2 SYNTHETIC ANTINEOPLASTIC AGENTS DERIVED FROM DOLASTATIN 15 AND METHODS OF MAKING SAME ARIZONA BOARD OF REGENTS (US) 2000-11-08 EP disclosed
WO-1999015130-A2 SYNTHETIC ANTINEOPLASTIC AGENTS DERIVED FROM DOLASTATIN 15 AND METHODS OF MAKING SAME ARIZONA BOARD OF REGENTS, actingon behalf of ARIZ ONA STATE UNIVERSITY (US) 1999-04-01 WO disclosed