SCHEMBL6233459

SCHEMBL6233459

CC1=C(c2c(C)cccc2C(=O)N2Cc3ccc(C(=O)N4CCN(C)CC4)n3Cc3ccccc32)CCC[C@H]1O

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 13/20 0.48
AVPR1A P37288 6/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
OXTR P30559 1/20 0.33
C5AR1 P21730 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5143793 0.84 AVPR2 (0.46) AVPR2AVPR1AOXTR
SCHEMBL5111220 0.84 AVPR2 (0.46) AVPR2AVPR1AOXTR
SCHEMBL5119243 0.84 AVPR2 (0.46) AVPR2AVPR1AOXTR
SCHEMBL6191112 0.81 AVPR2 (0.45) AVPR2AVPR1AOXTR
SCHEMBL5105261 0.81 AVPR2 (0.45) AVPR2AVPR1AOXTR
SCHEMBL5119149 0.75 AVPR2 (0.49) AVPR2AVPR1AKMT2AOXTR
SCHEMBL5117311 0.73 AVPR2 (0.43) AVPR2AVPR1A
SCHEMBL5117936 0.73 AVPR2 (0.43) AVPR2AVPR1A
SCHEMBL5785129 0.72 AVPR2 (0.61) AVPR2AVPR1A
SCHEMBL5628972 0.71 AVPR2 (0.48) AVPR2AVPR1AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1377585-B1 NOVEL 10-CYCLOHEXENYL-PHENYL PYRROLOBENZODIAZEPINE-3-CARBOXAMIDES AND DERIVATIVES THEREOF; TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS WYETH CORP (US) 2005-11-09 EP claimed