SCHEMBL6233751

SCHEMBL6233751

COc1cc(-c2ccc3c(c2)Nc2ccc(OC(C)=O)cc2NC3=O)ccc1O

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 19/20 0.70
AURKB Q96GD4 6/20 0.65
PIM1 P11309 5/20 0.65
CDK5 Q00535 5/20 0.65
TAOK1 Q7L7X3 5/20 0.65
MAP4K4 O95819 4/20 0.65
GSK3A P49840 4/20 0.65
PRKX P51817 4/20 0.65
PDPK1 O15530 3/20 0.65
CHEK2 O96017 3/20 0.65
CDK1 P06493 3/20 0.65
CDK2 P24941 3/20 0.65
GSK3B P49841 3/20 0.65
CAMK2D Q13557 3/20 0.65
PBK Q96KB5 3/20 0.65
STK17A Q9UEE5 3/20 0.65
MAP4K5 Q9Y4K4 3/20 0.65
CDK9 P50750 3/20 0.65
CDK8 P49336 3/20 0.65
PRKAA1 Q13131 3/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16712613 0.94 CHEK1 (0.70) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL6234226 0.85 CHEK1 (0.72) CHEK1
SCHEMBL4852172 0.83 CHEK1 (0.80) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL4860069 0.83 CHEK1 (1.00) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL4849727 0.83 CHEK1 (0.73) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL4854888 0.82 CHEK1 (0.69) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL4849157 0.82 CHEK1 (0.72) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL4858729 0.81 CHEK1 (0.78) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL4850212 0.81 CHEK1 (0.73) CHEK1AURKBPIM1CDK5TAOK1
SCHEMBL4858765 0.80 CHEK1 (0.69) CHEK1AURKBPIM1CDK5TAOK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1606268-A1 HETEROCYCLIC KINASE INHIBITORS Abbott Laboratories (US) 2005-12-21 EP claimed
WO-2004076424-A1 HETEROCYCLIC KINASE INHIBITORS ABBOTT LABORATORIES (US) 2004-09-10 WO claimed