SCHEMBL6233839

SCHEMBL6233839

Cn1c(N2CC[C@H](O)C2)nc2ccc(N)cc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 1/20 0.38
CDK2 P24941 1/20 0.38
PDE10A Q9Y233 1/20 0.37
HRH4 Q9H3N8 1/20 0.36
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
OPRK1 P41145 2/20 0.35
OGFRL1 Q5TC84 2/20 0.35
IKBKB O14920 2/20 0.35
GRM1 Q13255 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HTT P42858 1/20 0.35
MAPT P10636 2/20 0.34
SHMT2 P34897 1/20 0.34
IRAK1 P51617 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
CYP3A4 P08684 1/20 0.34
HTR2B P41595 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25599107 0.82 KDM4E (0.42) CDK2IKBKBALDH1A1HTTMAPT
SCHEMBL31349416 0.76 MAPT (0.51) ALDH1A1MAPTHPGD
SCHEMBL14824462 0.76 MAPT (0.51) ALDH1A1MAPTHPGD
SCHEMBL17487739 0.75 KCNH2 (0.43) ALDH1A1HPGDCNR2TRPC6
SCHEMBL3577361 0.71 MCHR1 (0.44) PDE10AMAPTHTR2B
SCHEMBL31349362 0.70 BRD4 (0.36) GRM1ALDH1A1MAPTCYP3A4HTR2B
SCHEMBL3251853 0.70 MAPT (0.57) CDK1CDK2PDE10AALDH1A1HTT
SCHEMBL18960406 0.69 CHEK2 (0.43) HRH4
SCHEMBL18344077 0.69 NPC1 (0.47) CDK1CDK2PDE10AALDH1A1MAPT
SCHEMBL18344021 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004092181-A9 HETEROCYCLIC MCHR1 ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2005-01-27 WO disclosed