SCHEMBL6237575

SCHEMBL6237575

Nc1c(Cl)ncnc1Nc1ccc(F)c(Cl)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.64
GRM1 Q13255 1/20 0.61
MAPK1 P28482 1/20 0.58
ERBB2 P04626 2/20 0.55
KDR P35968 4/20 0.53
AURKA O14965 2/20 0.53
FBP1 P09467 2/20 0.53
INSR P06213 1/20 0.53
PDGFRB P09619 1/20 0.53
FLT4 P35916 1/20 0.53
CLK1 P49759 1/20 0.53
EPHB4 P54760 1/20 0.53
TEK Q02763 1/20 0.53
AURKB Q96GD4 1/20 0.53
RPS6KB1 P23443 1/20 0.52
BRAF P15056 1/20 0.50
POLB P06746 1/20 0.50
MAPT P10636 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
DYRK1A Q13627 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17815581 0.81 EGFR (0.49) EGFRAURKAMAPTSMN1; SMN2
SCHEMBL1896427 0.81 TTBK1 (0.55) EGFRKDRMAPT
SCHEMBL4274133 0.79 EGFR (0.55) EGFRGRM1MAPK1ERBB2KDR
SCHEMBL3061494 0.79 EGFR (0.62) EGFRMAPK1ERBB2FBP1PDGFRB
SCHEMBL30683235 0.78 EGFR (0.59) EGFRGRM1MAPK1ERBB2KDR
SCHEMBL26618910 0.78 EGFR (0.59) EGFRGRM1MAPK1ERBB2KDR
SCHEMBL31299934 0.78 EGFR (1.00) EGFRGRM1ERBB2KDRAURKA
SCHEMBL1096688 0.78 EGFR (0.60) EGFRGRM1MAPK1ERBB2KDR
SCHEMBL8311292 0.78 EGFR (0.77) EGFRGRM1ERBB2KDRAURKA
SCHEMBL19762918 0.78 EGFR (0.69) EGFRGRM1MAPK1ERBB2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005009384-A2 EGFR TYROSINE KINASE INHIBITORS IMCLONE SYSTEMS INCORPORATED (US) 2005-02-03 WO disclosed